SCHEMBL10522115

SCHEMBL10522115

O=C1CC2CCCCN2C=N1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTDSP1 Q9GZU7 1/20 0.46
ALDH1A1 P00352 3/20 0.31
PKM P14618 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5447508 0.73 ALDH1A1 (0.36) CTDSP1ALDH1A1PKMSMN1; SMN2CYP3A4
SCHEMBL2919397 0.66
SCHEMBL5421843 0.64 ALDH1A1 (0.31) ALDH1A1SMN1; SMN2CYP3A4CYP2C9CYP2C19
SCHEMBL7491125 0.64
SCHEMBL7490975 0.63
SCHEMBL2114822 0.62 CTDSP1 (0.49) CTDSP1ALDH1A1SMN1; SMN2CYP3A4CYP2C9
SCHEMBL4462216 0.61
SCHEMBL9265060 0.59
SCHEMBL7488301 0.59
SCHEMBL22651958 0.59

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4791199-A Process for antiarrhythmic 1,3-diazabicyclo[4.4.0]dec-2-en-4-ones G. D. SEARLE & CO. (US) 1988-12-13 US claimed
EP-0215477-A1 Process and intermediates for antiarrhytmic 1,3-diazabicyclo/4.4.0/dec-2-en-4-ones G.D. Searle & Co. (US) 1987-03-25 EP claimed
EP-0175319-B1 HEXAHYDROINDOLIZINONES G.D. Searle & Co. (US) 1989-12-06 EP disclosed
US-4791199-A Process for antiarrhythmic 1,3-diazabicyclo[4.4.0]dec-2-en-4-ones G. D. SEARLE & CO. (US) 1988-12-13 US disclosed
US-4791199-A Process for antiarrhythmic 1,3-diazabicyclo[4.4.0]dec-2-en-4-ones G. D. SEARLE & CO. (US) 1988-12-13 US disclosed
US-4791199-A Process for antiarrhythmic 1,3-diazabicyclo[4.4.0]dec-2-en-4-ones G. D. SEARLE & CO. (US) 1988-12-13 US disclosed
EP-0104647-B1 PYRIDOPYRIMIDINONES G.D. Searle & Co. (US) 1988-03-30 EP disclosed
EP-0234331-A1 Octahydropyrido[1,2-c]-pyrimidinones G.D. Searle & Co. (US) 1987-09-02 EP disclosed
US-4680295-A ANTIARRHYTHMIA AGENTS G. D. SEARLE & CO. (US) 1987-07-14 US disclosed
EP-0215477-A1 Process and intermediates for antiarrhytmic 1,3-diazabicyclo/4.4.0/dec-2-en-4-ones G.D. Searle & Co. (US) 1987-03-25 EP disclosed
EP-0215477-A1 Process and intermediates for antiarrhytmic 1,3-diazabicyclo/4.4.0/dec-2-en-4-ones G.D. Searle & Co. (US) 1987-03-25 EP disclosed
EP-0215477-A1 Process and intermediates for antiarrhytmic 1,3-diazabicyclo/4.4.0/dec-2-en-4-ones G.D. Searle & Co. (US) 1987-03-25 EP disclosed
EP-0175319-A1 Hexahydroindolizinones G.D. Searle & Co. (US) 1986-03-26 EP disclosed
US-4567270-A Hexahydroindolizinones useful for treating cardiac arrhythmia, thrombotic disorders in mammals G. D. SEARLE & CO. (US) 1986-01-28 US disclosed
US-4560754-A Substituted 5-phenyl-5-(aminoalkyl)-1,3-diazabicyclo[4.4.0]decan-4-ones and 5-phenyl-5-(aminoalkyl)-1,3-diazabicyclo[4.4.0]dec-2-en-4-ones G. D. SEARLE & CO. (US) 1985-12-24 US disclosed