SCHEMBL105276

SCHEMBL105276

CN(C)CCNC(=O)c1cccc2cc3ccccc3nc12

nearest known ligand 0.78

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AOX1 Q06278 1/20 0.78
RAD52 P43351 7/20 0.69
UHRF1 Q96T88 2/20 0.65
SMARCA2 P51531 1/20 0.63
HDAC1 Q13547 1/20 0.63
HDAC6 Q9UBN7 1/20 0.63
ALDH1A1 P00352 3/20 0.53
KDM4E B2RXH2 2/20 0.53
HSD17B10 Q99714 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
POLR1A O95602 2/20 0.52
ECE1 P42892 1/20 0.52
MUS81 Q96NY9 1/20 0.52
HTT P42858 1/20 0.51
HTR2C P28335 1/20 0.50
MOK Q9UQ07 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29369424 1.00 AOX1 (0.78) AOX1RAD52UHRF1SMARCA2HDAC1
Hydrochloric Acid SCHEMBL29608361 0.99 AOX1 (0.77) AOX1RAD52UHRF1SMARCA2HDAC1
Hydrochloric Acid SCHEMBL4888175 0.99 AOX1 (0.77) AOX1RAD52UHRF1SMARCA2HDAC1
Hydrochloric Acid SCHEMBL5953779 0.97 AOX1 (0.75) AOX1RAD52UHRF1SMARCA2HDAC1
SCHEMBL8711841 0.94 AOX1 (0.71) AOX1RAD52UHRF1SMARCA2HDAC1
SCHEMBL7023521 0.88 AOX1 (0.69) AOX1RAD52UHRF1SMARCA2HDAC1
SCHEMBL7032809 0.88 AOX1 (0.69) AOX1RAD52UHRF1SMARCA2HDAC1
SCHEMBL2447168 0.88 KDM4E (0.69) AOX1RAD52UHRF1SMARCA2HDAC1
SCHEMBL7566347 0.88 HDAC1 (0.67) AOX1RAD52UHRF1SMARCA2HDAC1
SCHEMBL7024435 0.87 AOX1 (0.74) AOX1RAD52UHRF1SMARCA2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2684 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144882-A1 ANTI-NECTIN-4 ANTIBODY DRUG CONJUGATE AND USE THEREOF BIO-THERA SOLUTIONS, LTD. (CN) 2026-05-28 US claimed
US-20260008848-A1 ANTI-NECTIN-4 ANTIBODY, AND ANTIBODY-DRUG CONJUGATE AND USE THEREOF BIO THERA SOLUTIONS LTD (CN) 2026-01-08 US claimed
US-20250381283-A1 METHOD FOR TREATING SOLID TUMOR BIO THERA SOLUTIONS LTD (CN) 2025-12-18 US claimed
US-20250333498-A1 ANTI-CLDN18.2 ANTIBODY, AND ANTIBODY-DRUG CONJUGATE AND USE THEREOF BIO THERA SOLUTIONS LTD (CN) 2025-10-30 US claimed
US-20250262316-A1 ANTIBODY-DRUG CONJUGATE AND APPLICATION THEREOF BIO-THERA SOLUTIONS, LTD. (CN) 2025-08-21 US claimed
US-20250249114-A1 METHOD FOR TREATING HER2-POSITIVE SOLID TUMOR BIO-THERA SOLUTIONS, LTD. (CN) 2025-08-07 US claimed
EP-4556027-A1 ANTI-NECTIN-4 ANTIBODY DRUG CONJUGATE AND USE THEREOF Bio-Thera Solutions, Ltd. (CN) 2025-05-21 EP claimed
EP-4545099-A1 METHOD FOR TREATING SOLID TUMOR Bio-Thera Solutions, Ltd. (CN) 2025-04-30 EP claimed
EP-4538291-A1 ANTI-NECTIN-4 ANTIBODY, AND ANTIBODY-DRUG CONJUGATE AND USE THEREOF Bio-Thera Solutions, Ltd. (CN) 2025-04-16 EP claimed
EP-4534105-A1 ANTI-CLDN18.2 ANTIBODY, AND ANTIBODY-DRUG CONJUGATE AND USE THEREOF Bio-Thera Solutions, Ltd. (CN) 2025-04-09 EP claimed
WO-2002085459-A2 ANTIANGIOGENIC COMBINATION THERAPY FOR THE TREATMENT OF CANCER PHARMACIA CORPORATION (US) 2002-10-31 WO claimed
US-20020103141-A1 Antiangiogenic combination therapy for the treatment of cancer PHARMACIA CORPORATION 2002-08-01 US claimed
EP-0642343-B1 Acridine carboxamides for the treatment of cancer XENOVA LTD (GB) 2000-08-30 EP claimed
US-6111109-A CYCLIZING A 2-(2-ALKYLOXYCARBONYLPHENYL)AMINO-)BENZALDEHYDE BY TREATING WITH A BORON TRIFLUORIDE; NEUTRALIZATION OF THE FORMED SALT; AMIDATION WITH AN 2-N,N-DIALKYLAMINOETHYLAMINE;ANTITUMOR AND -CARCINOGENIC XENOVA LIMITED (GB) 2000-08-29 US claimed
EP-0934277-A1 PROCESS FOR THE PREPARATION OF N- 2-(DIMETHYLAMINO)ETHYL]ACRIDINE-4-CARBOXAMIDE XENOVA LIMITED (GB) 1999-08-11 EP claimed
US-5891886-A PREVENTION DRUG RESISTANCE; ADMINISTERING N-(2-(DIMETHYLAMINO)ETHYL)ACRIDINE-4-CARBOXAMIDE XENOVA LIMITED (GB) 1999-04-06 US claimed
WO-1998017649-A1 PROCESS FOR THE PREPARATION OF N-[2-(DIMETHYLAMINO)ETHYL]ACRIDINE-4-CARBOXAMIDE XENOVA LIMITED (GB) 1998-04-30 WO claimed
US-5696131-A ADMINISTERING N-(2-(DIMETHYLAMINO)ETHYL)ACRIDINE-4-CARBOXAMIDE WITH OTHER ANTICANCER DRUGS IN A DIVIDED-DOSE SCHEDULE XENOVA LIMITED (GB) 1997-12-09 US claimed
EP-0642343-A1 TREATMENT OF CANCERS XENOVA LIMITED (GB) 1995-03-15 EP claimed
WO-1993024096-A2 USE OF N-(2-(DIMETHYLAMINO)ETHYL)ACRIDINE-4-CARBOXAMIDE AND ITS ANALOGUES FOR CANCER TREATMENT XENOVA LIMITED (GB) 1993-12-09 WO claimed