SCHEMBL10528142

SCHEMBL10528142

Cc1cc(C(C)CCC2CCCCC2)c(C)cn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LNPEP Q9UIQ6 3/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
ALOX5 P09917 2/20 0.32
PTGES O14684 1/20 0.32
PTGS2 P35354 1/20 0.32
PPARG P37231 1/20 0.32
PSEN1 P49768 1/20 0.32
ALDH1A1 P00352 1/20 0.31
LCK P06239 1/20 0.31
KIT P10721 1/20 0.31
SRC P12931 1/20 0.31
KDR P35968 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10527380 0.77 OPRL1 (0.44) NPC1MEN1TP53TSHRRAB9A
SCHEMBL10525803 0.77 CDK1 (0.33) LNPEP
SCHEMBL10528028 0.76 ADRB2 (0.39) TSHRALDH1A1GAAHTT
SCHEMBL21711087 0.75 UHRF1 (0.35)
SCHEMBL10528162 0.74 NPC1 (0.42) NPC1MEN1TP53TSHRRAB9A
SCHEMBL10525949 0.74 SMN1; SMN2 (0.35) TSHRRAB9ASMN1; SMN2LNPEPALDH1A1
SCHEMBL10529845 0.74 RAB9A (0.38) NPC1MEN1TP53TSHRRAB9A
SCHEMBL10525897 0.73 NPC1 (0.35) NPC1MEN1TP53TSHRRAB9A
SCHEMBL10528254 0.73 OPRL1 (0.36) NPC1MEN1TP53TSHRRAB9A
SCHEMBL10529833 0.71 TSHR (0.40) NPC1MEN1TP53TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0253681-A2 Cycloalkyl-substituted 4-pyridyl derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-01-20 EP claimed
US-4797411-A ANTITUMOR AGENTS FARMITALIA CARLO ERBA S.P.A. (IT) 1989-01-10 US disclosed
EP-0253681-A2 Cycloalkyl-substituted 4-pyridyl derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-01-20 EP disclosed