SCHEMBL10529622

SCHEMBL10529622

NS(=O)(=O)c1ccc(SCCCO)c([N+](=O)[O-])c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA2 P00918 14/20 1.00
ALDH1A1 P00352 1/20 0.56
CA12 O43570 3/20 0.54
CA1 P00915 3/20 0.54
CA9 Q16790 3/20 0.54
VCAM1 P19320 1/20 0.49
GSTP1 P09211 3/20 0.47
GSTM2 P28161 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10528943 0.92 CA2 (1.00) CA2ALDH1A1CA12CA1CA9
SCHEMBL6114282 0.80 CA2 (0.70) CA2ALDH1A1CA12CA1CA9
SCHEMBL2831588 0.77 CA2 (0.66) CA2ALDH1A1CA12CA1CA9
SCHEMBL9877839 0.77 CA2 (0.73) CA2ALDH1A1GSTP1GSTM2SMN1; SMN2
SCHEMBL10528739 0.77 CA2 (1.00) CA2CA12CA1CA9
SCHEMBL1700058 0.76 CA2 (0.64) CA2ALDH1A1CA12CA1CA9
SCHEMBL10528804 0.74 CA2 (0.66) CA2CA12CA1CA9VCAM1
SCHEMBL10529657 0.73 CA2 (1.00) CA2ALDH1A1
SCHEMBL11876450 0.73 CA2 (0.68) CA2ALDH1A1GSTP1GSTM2
SCHEMBL6851577 0.71 MAPT (0.66) CA2ALDH1A1CA12CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0219429-B1 SUBSTITUTED BENZENESULFONAMIDE AND ANTIGLAUCOMA FORMULATIONS CONTAINING THEM MERCK & CO. INC. (US) 1989-12-20 EP disclosed
US-4678855-A CARBONIC ANHYDRASE INHIBITORS, GLAUCOMA MERCK & CO., INC. (US) 1987-07-07 US disclosed
EP-0219429-A1 Substituted benzenesulfonamide and antiglaucoma formulations containing them MERCK & CO. INC. (US) 1987-04-22 EP disclosed