SCHEMBL10539689

SCHEMBL10539689

N#C[CH]C(=O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.55
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
TSHR P16473 1/20 0.52
ALDH1A1 P00352 1/20 0.52
MAPK1 P28482 1/20 0.52
CYP1B1 Q16678 1/20 0.51
MAPT P10636 1/20 0.50
RAB9A P51151 1/20 0.50
MAOB P27338 5/20 0.49
MAOA P21397 3/20 0.49
CES2 O00748 1/20 0.49
SRD5A2 P31213 1/20 0.49
BCHE P06276 1/20 0.47
GSK3B P49841 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL836819 0.79 CES1 (0.61) CES1CA1CA2TDP1TSHR
SCHEMBL10541210 0.78 CES1 (0.50) CES1CA1CA2TDP1TSHR
SCHEMBL360287 0.77 CES1 (0.63) CES1CA1CA2TDP1TSHR
SCHEMBL7918197 0.76 CES1 (0.61) CES1CA1CA2TDP1TSHR
SCHEMBL5099884 0.76 CES1 (0.61) CES1CA1CA2TDP1TSHR
SCHEMBL8024786 0.76 MAPK1 (0.62) CES1CA1CA2TDP1TSHR
SCHEMBL10861302 0.74 TDP1 (0.62) CES1CA1CA2TDP1TSHR
SCHEMBL6230475 0.74 ALDH1A1 (0.55) CES1CA1CA2TDP1TSHR
SCHEMBL6230478 0.74 ALDH1A1 (0.55) CES1CA1CA2TDP1TSHR
SCHEMBL6230468 0.74 ALDH1A1 (0.55) CES1CA1CA2TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4829076-A CARDIOVASCULAR DISORDERS ALKALOIDA VEGYESZETI GYAR (HU) 1989-05-09 US disclosed