SCHEMBL10539706

SCHEMBL10539706

O=C(c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1)c1cc(Cl)cc2c1OCOC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.41
USP2 O75604 2/20 0.41
ALDH1A1 P00352 4/20 0.38
KMT2A Q03164 3/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
GAA P10253 2/20 0.38
HPGD P15428 2/20 0.38
MEN1 O00255 1/20 0.38
NPSR1 Q6W5P4 2/20 0.35
PKM P14618 1/20 0.35
CXCR5 P32302 1/20 0.34
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
ENPP2 Q13822 1/20 0.33
KDM4E B2RXH2 3/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10539494 0.82 SIRT2 (0.32) ENPP2
SCHEMBL9521500 0.78 TSHR (0.41) TSHRUSP2ALDH1A1KMT2ANPC1
SCHEMBL9521480 0.77 TSHR (0.40) TSHRUSP2ALDH1A1KMT2ANPC1
SCHEMBL31298404 0.74 PARP1 (0.47) NPSR1MAPTENPP2HCRTR1HCRTR2
SCHEMBL5682164 0.73 CYP11B1 (0.43) KMT2AENPP2CYP1A2
SCHEMBL3752469 0.72 HCRTR1 (0.40) USP2KMT2AMEN1MAPTENPP2
SCHEMBL23879944 0.69 ALDH1A1 (0.43) TSHRUSP2ALDH1A1KMT2ANPC1
SCHEMBL693097 0.69 CYP11B1 (0.41) TSHRUSP2KMT2ARAB9AMEN1
SCHEMBL670904 0.68 CYP11B1 (0.43) TSHRALDH1A1HPGDENPP2KDM4E
SCHEMBL9518291 0.68 TSHR (0.35) TSHRUSP2ALDH1A1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4816452-A ANTIBIOTICS BEECHAM GROUP P.L.C. (GB) 1989-03-28 US disclosed
US-4814343-A ANTIISCHEMIC U C B, S.A. (BE) 1989-03-21 US disclosed
EP-0210815-A2 6-Beta-(alpha-etherified oxyimino)-acylamino penicillanic-acid derivatives, their preparation and use BEECHAM GROUP PLC (GB) 1987-02-04 EP disclosed