SCHEMBL10550202

SCHEMBL10550202

CCOC(=O)c1cc(F)c(O)nc1Nc1ccc(F)cc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.53
TSHR P16473 3/20 0.48
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
MAP2K2 P36507 1/20 0.44
MAP2K1 Q02750 1/20 0.44
MAPK14 Q16539 1/20 0.44
LMNA P02545 3/20 0.42
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 1/20 0.42
ALPL P05186 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
POLB P06746 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TRPM8 Q7Z2W7 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10546863 0.88 NPC1 (0.45) THRBHTTMAPK14LMNAMAPT
SCHEMBL10548932 0.87 THRB (0.46) THRBTSHRMAPK1HTTMAPK14
SCHEMBL10757185 0.81 CSNK2A1 (0.47) HTTMAP2K2MAP2K1LMNAMAPT
SCHEMBL10467490 0.79 KDM4E (0.48) TSHRMAPTNPC1ALDH1A1HPGD
SCHEMBL10550001 0.79 THRB (0.44) THRBHTTMAPK14LMNAMAPT
SCHEMBL10469421 0.78 KDM4E (0.43) TSHRLMNASMN1; SMN2ALDH1A1GAA
SCHEMBL10547734 0.77 THRB (0.45) THRBTSHRMAPK14LMNAMAPT
SCHEMBL10467363 0.76 ALDH1A1 (0.47) TSHRMAPK1HTTLMNAMAPT
SCHEMBL10549993 0.76 NPC1 (0.43) THRBHTTLMNAMAPTSMN1; SMN2
SCHEMBL10548728 0.76 THRB (0.44) THRBTSHRMAPK14MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4851535-A 2-(5-FLUORONICOTINOYL)ACETIC ACID DERIVATIVES, ANTIBACTERIAL 1-ARYL-1,4-DIHYDRO-4-OXONAPHTHYRIDINES TOYAMA CHEMICAL CO., LTD. (JP) 1989-07-25 US disclosed
US-4704459-A VILSMEIER REAGENT TOYAMA CHEMICAL CO., LTD. (JP) 1987-11-03 US disclosed