SCHEMBL10550681

SCHEMBL10550681

CCOC(=O)c1cn(-c2ccc(F)cc2F)c2nc(OS(=O)(=O)c3ccccc3[N+](=O)[O-])c(F)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
MAPT P10636 5/20 0.43
LMNA P02545 3/20 0.43
NPC1 O15118 1/20 0.41
POLB P06746 3/20 0.40
KDM4E B2RXH2 3/20 0.40
HPGD P15428 3/20 0.40
HSD17B10 Q99714 3/20 0.40
HTT P42858 2/20 0.40
XBP1 P17861 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
KMT2A Q03164 2/20 0.39
EPHA2 P29317 1/20 0.38
FLT4 P35916 1/20 0.38
GSK3B P49841 1/20 0.38
RARB P10826 1/20 0.38
TBXAS1 P24557 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10550405 0.83 ALDH1A1 (0.43) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL10549552 0.81 KMT2A (0.47) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL10551019 0.80 ALDH1A1 (0.40) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL5416374 0.78 KMT2A (0.52) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL10549291 0.78 KMT2A (0.49) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL10550253 0.78 ALDH1A1 (0.47) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL10548813 0.78 ALDH1A1 (0.46) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL10549467 0.77 KMT2A (0.43) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL10549101 0.77 KMT2A (0.44) ALDH1A1MAPTLMNAPOLBKDM4E
SCHEMBL3236130 0.77 KMT2A (0.48) ALDH1A1MAPTLMNANPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4851535-A 2-(5-FLUORONICOTINOYL)ACETIC ACID DERIVATIVES, ANTIBACTERIAL 1-ARYL-1,4-DIHYDRO-4-OXONAPHTHYRIDINES TOYAMA CHEMICAL CO., LTD. (JP) 1989-07-25 US disclosed
US-4704459-A VILSMEIER REAGENT TOYAMA CHEMICAL CO., LTD. (JP) 1987-11-03 US disclosed