SCHEMBL10550802

SCHEMBL10550802

CC(C(=O)N1CCN(C)CC1)C1c2ccccc2C(=O)N1c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.52
HSD17B10 Q99714 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CHRM3 P20309 3/20 0.43
ALDH1A1 P00352 3/20 0.42
MAPT P10636 1/20 0.42
CHRM1 P11229 4/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
TSHR P16473 2/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10554431 0.89 ALDH1A1 (0.51) NPC1HSD17B10LMNAKMT2AMEN1
SCHEMBL10551223 0.81 GAA (0.49) NPC1HSD17B10LMNAKMT2AMEN1
SCHEMBL4124062 0.76 NPC1 (0.39) NPC1LMNAKMT2AMEN1CYP1A2
SCHEMBL10550805 0.74 KMT2A (0.54) HSD17B10LMNAKMT2AMEN1CYP1A2
SCHEMBL11162182 0.70 ALDH1A1 (0.49) NPC1HSD17B10LMNAKMT2AMEN1
SCHEMBL29874882 0.69 POLB (0.47) NPC1HSD17B10KMT2AMEN1CYP1A2
SCHEMBL30467237 0.68 POLB (0.46) NPC1HSD17B10LMNAKMT2AMEN1
SCHEMBL10554827 0.67 ALDH1A1 (0.48) NPC1KMT2AMEN1CYP1A2CYP3A4
SCHEMBL29538871 0.66 KMT2A (0.42) HSD17B10LMNAKMT2AMEN1CYP1A2
SCHEMBL11817121 0.65 HSD17B10 (0.50) NPC1HSD17B10CHRM3CHRM1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4879293-A NERVOUS SYSTEM AND PSYCHOSOMATIC DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-11-07 US disclosed
US-4788191-A ANTIANXIETY AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1988-11-29 US disclosed
US-4590189-A ANTIANXIETY AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1986-05-20 US disclosed