SCHEMBL10554135

SCHEMBL10554135

O=[N+]([O-])c1cc(CCN2CCCCC2)ccc1OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.61
HRH3 Q9Y5N1 2/20 0.55
HTR1A P08908 1/20 0.54
DRD2 P14416 1/20 0.54
HTR2A P28223 1/20 0.54
SIGMAR1 Q99720 6/20 0.50
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
CTSV O60911 1/20 0.47
CTSL P07711 1/20 0.47
SLC6A3 Q01959 1/20 0.47
HPGD P15428 2/20 0.45
LMNA P02545 1/20 0.45
LTA4H P09960 1/20 0.45
PTGS1 P23219 1/20 0.45
PTGS2 P35354 1/20 0.45
FAAH O00519 1/20 0.45
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10554521 1.00 POLB (0.61) POLBHRH3HTR1ADRD2HTR2A
SCHEMBL10556415 0.99 POLB (0.62) POLBHRH3HTR1ADRD2HTR2A
SCHEMBL10553527 0.84 POLB (0.53) POLBHTR1ADRD2HTR2AALDH1A1
SCHEMBL10551296 0.83 ALDH1A1 (0.55) POLBHTR1ADRD2HTR2AALDH1A1
SCHEMBL10556424 0.82 POLB (0.53) POLBHTR1ADRD2HTR2AALDH1A1
SCHEMBL18159251 0.82 HRH3 (0.55) HRH3HTR1ADRD2HTR2ASIGMAR1
SCHEMBL10553555 0.80 HRH3 (0.61) HRH3SIGMAR1MEN1KMT2ASLC6A3
SCHEMBL10555657 0.80 HRH3 (0.61) HRH3SIGMAR1MEN1KMT2ASLC6A3
SCHEMBL10553541 0.80 POLB (0.50) POLBALDH1A1MEN1KMT2ACTSV
SCHEMBL6814063 0.79 POLB (0.54) POLBHTR1AALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4847269-A GLAUCOMA, AMIDES OR UREA DERIVATIVES OF AMINOETHYLCARBOXY COMPOUNDS SYNTEX (U.S.A.) INC. (US) 1989-07-11 US disclosed
US-4629730-A ADMINISTERING DIALKYL OR CYCLOAKYL AMINO ETHYLANILINE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1986-12-16 US disclosed
EP-0180994-A2 Antihypertensive dialkyl aminoethylaniline derivatives SYNTEX (U.S.A.) INC. (US) 1986-05-14 EP disclosed