SCHEMBL10554346

SCHEMBL10554346

O=CNc1cc(CCN2CCCCCC2)ccc1OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.54
SIGMAR1 Q99720 3/20 0.49
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SLC6A3 Q01959 1/20 0.46
MET P08581 1/20 0.45
APP P05067 1/20 0.43
LTA4H P09960 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
EPHX2 P34913 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
NPY1R P25929 1/20 0.42
EGFR P00533 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10553207 1.00 HRH3 (0.54) HRH3SIGMAR1MEN1KMT2ASLC6A3
SCHEMBL10555526 0.99 HRH3 (0.55) HRH3SIGMAR1MEN1KMT2ASLC6A3
SCHEMBL10557212 0.85 HTR6 (0.40) HRH3SIGMAR1MEN1KMT2AALDH1A1
SCHEMBL10923941 0.83 SIGMAR1 (0.54) HRH3SIGMAR1MEN1KMT2AMET
SCHEMBL10922973 0.83 SIGMAR1 (0.54) HRH3SIGMAR1MEN1KMT2AMET
SCHEMBL10551022 0.83 KDM4E (0.39) HRH3SIGMAR1MEN1KMT2AKDM4E
SCHEMBL10555532 0.83 FFAR4 (0.40) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL10554118 0.83 BRD4 (0.56) HRH3SIGMAR1MEN1KMT2AMET
Bromide SCHEMBL10552937 0.83 SIGMAR1 (0.53) HRH3SIGMAR1MEN1KMT2AMET
SCHEMBL10554709 0.83 BRD4 (0.56) HRH3SIGMAR1MEN1KMT2AMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4847269-A GLAUCOMA, AMIDES OR UREA DERIVATIVES OF AMINOETHYLCARBOXY COMPOUNDS SYNTEX (U.S.A.) INC. (US) 1989-07-11 US disclosed
US-4629730-A ADMINISTERING DIALKYL OR CYCLOAKYL AMINO ETHYLANILINE DERIVATIVES SYNTEX (U.S.A.) INC. (US) 1986-12-16 US disclosed
EP-0180994-A2 Antihypertensive dialkyl aminoethylaniline derivatives SYNTEX (U.S.A.) INC. (US) 1986-05-14 EP disclosed