SCHEMBL10558762

SCHEMBL10558762

O=C(Nc1cccc(Cn2ccnc2)c1)c1ccccn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.56
CYP19A1 P11511 2/20 0.55
KDR P35968 6/20 0.55
GRM4 Q14833 2/20 0.54
HDAC6 Q9UBN7 1/20 0.54
KCNK3 O14649 1/20 0.53
KCNK9 Q9NPC2 1/20 0.53
ACKR3 P25106 1/20 0.52
CYP11B1 P15538 4/20 0.52
CYP11B2 P19099 4/20 0.52
CYP1A2 P05177 1/20 0.52
POLB P06746 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
MAPT P10636 1/20 0.52
TBXAS1 P24557 1/20 0.52
QPCT Q16769 1/20 0.52
CYP4Z1 Q86W10 1/20 0.52
QPCTL Q9NXS2 1/20 0.52
AGTR2 P50052 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10465391 0.87 MAPT (0.52) S1PR1CYP19A1CYP11B1CYP11B2CYP1A2
Hydrochloric Acid SCHEMBL10464770 0.85 MAPT (0.50) S1PR1CYP19A1CYP11B1CYP11B2CYP1A2
SCHEMBL24449229 0.84 ACKR3 (0.54) S1PR1CYP19A1ACKR3CYP11B1CYP11B2
SCHEMBL13604350 0.82 MEN1 (0.63) CYP19A1CYP11B1CYP11B2CYP1A2POLB
SCHEMBL15014091 0.77 GRM4 (0.65) KDRGRM4HDAC6KCNK3KCNK9
SCHEMBL7990375 0.76 KDR (0.84) KDRGRM4HDAC6KCNK3KCNK9
SCHEMBL4486676 0.76 AGTR2 (0.52) S1PR1CYP19A1CYP11B1CYP11B2TBXAS1
SCHEMBL31610004 0.75 NPC1 (0.58) CYP19A1POLBTBXAS1
SCHEMBL13006757 0.74 CYP11B1 (0.66) CYP19A1CYP11B1CYP11B2CYP1A2POLB
SCHEMBL13153532 0.74 GRM4 (0.60) KDRGRM4HDAC6KCNK3KCNK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4873238-A ANTIULCER AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1989-10-10 US disclosed