SCHEMBL10560352

SCHEMBL10560352

CC(=O)Nc1ccc(OCCCN2CCC(C(c3ccc(F)cc3)c3ccc(F)cc3)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.58
DRD2 P14416 5/20 0.58
HTR1A P08908 4/20 0.58
ADRA2A P08913 2/20 0.58
ADRA1D P25100 2/20 0.58
HTR2C P28335 2/20 0.58
ADRA1A P35348 2/20 0.58
HRH1 P35367 2/20 0.58
ADRA1B P35368 2/20 0.58
HTR6 P50406 2/20 0.58
KCNH2 Q12809 2/20 0.58
HRH3 Q9Y5N1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL10559966 0.99 HTR2A (0.57) HTR2ADRD2HTR1AADRA2AADRA1D
SCHEMBL10559681 0.91 DRD2 (0.55) HTR2ADRD2HTR1AADRA2AADRA1D
SCHEMBL10560816 0.87 HRH2 (0.58) HTR2AHRH1HRH3
SCHEMBL10460536 0.86 HTR2A (0.58) HTR2ADRD2HTR1AHRH1HRH3
Fumaric Acid SCHEMBL10461972 0.85 DRD2 (0.49) HTR2ADRD2HTR1AADRA2AADRA1D
Fumaric Acid SCHEMBL10461968 0.85 DRD2 (0.49) HTR2ADRD2HTR1AADRA2AADRA1D
SCHEMBL10558384 0.83 HTR2A (0.53) HTR2ADRD2HTR1AHRH3
Water SCHEMBL10557406 0.83 HTR2A (0.49) HTR2ADRD2HTR1AHRH1HRH3
SCHEMBL10556073 0.82 HRH3 (0.55) HTR2ADRD2HTR1AHRH1HRH3
Oxalic Acid SCHEMBL10461397 0.82 KDM4E (0.58) HTR2ADRD2HTR1AHRH1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4810713-A Arylalkyl-heterocyclic amines, n-substituted by aryloxyalkyl groups used in a method for allergy treatment A. H. ROBINS COMPANY, INCORPORATED (US) 1989-03-07 US claimed
EP-0235463-A2 N-substituted-arylalkyl and arylalkylene piperidines as cardiovascular antihistaminic and antisecretory agents A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1987-09-09 EP claimed