SCHEMBL10565622

SCHEMBL10565622

CC(C(c1ccc(OC(F)(F)F)cc1)c1ccc(OC(F)(F)F)cc1)n1cncn1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.44
CYP19A1 P11511 12/20 0.41
ALDH1A1 P00352 1/20 0.38
NPBWR1 P48145 1/20 0.38
MCHR1 Q99705 1/20 0.38
POLB P06746 1/20 0.38
HSP90AA1 P07900 1/20 0.38
CYP3A4 P08684 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CYP11B1 P15538 1/20 0.36
TSHR P16473 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP2C19 P33261 1/20 0.36
SCN5A Q14524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10564644 0.82 CYP19A1 (0.46) PDE2ACYP19A1HSP90AA1CYP3A4CYP11B1
SCHEMBL10565254 0.77 CYP19A1 (0.65) CYP19A1POLBHSP90AA1CYP3A4MEN1
SCHEMBL10565684 0.77 CYP19A1 (0.40) PDE2ACYP19A1NPBWR1MCHR1POLB
SCHEMBL10567440 0.76 CYP17A1 (0.46) PDE2ACYP19A1ALDH1A1NPBWR1MCHR1
SCHEMBL10565630 0.76 PDE2A (0.40) PDE2ACYP19A1ALDH1A1NPBWR1MCHR1
SCHEMBL9467692 0.76 POLB (0.38) PDE2ACYP19A1ALDH1A1POLBHSP90AA1
SCHEMBL9362897 0.76 CYP19A1 (0.43) CYP19A1ALDH1A1POLBHSP90AA1CYP3A4
SCHEMBL9467685 0.76 POLB (0.38) PDE2ACYP19A1ALDH1A1POLBHSP90AA1
SCHEMBL6947959 0.76 MEN1 (0.46) CYP19A1ALDH1A1POLBHSP90AA1CYP3A4
SCHEMBL10565696 0.75 CYP19A1 (0.41) PDE2ACYP19A1ALDH1A1NPBWR1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0194064-A2 Azolyl substituted aralkyl compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-09-10 EP claimed
US-4829074-A INSECTICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-09 US disclosed
EP-0194064-A2 Azolyl substituted aralkyl compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-09-10 EP disclosed