SCHEMBL10567702

SCHEMBL10567702

O=C(O)C1CCCN2C(=O)C[C@H](N3C(=O)c4ccccc4C3=O)C(=O)N12

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACE P12821 7/20 0.53
MME P08473 3/20 0.45
HSD17B10 Q99714 1/20 0.38
ALDH1A1 P00352 4/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
CHRM2 P08172 1/20 0.36
OPRM1 P35372 1/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
IKZF3 Q9UKT9 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5158143 0.89 ACE (0.51) ACEMMEHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL5154520 0.89 ACE (0.51) ACEMMEHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL5154528 0.89 ACE (0.51) ACEMMEHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL5154165 0.89 ACE (0.51) ACEMMEHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL5154587 0.89 ACE (0.51) ACEMMEHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL10561930 0.85 CASP3 (0.39) ACEMMEHSD17B10ALDH1A1DDB1
SCHEMBL644661 0.84 ACE (0.49) ACEMMEHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL6527218 0.84 ACE (0.47) ACEMMEHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL10565346 0.84 ACE (0.47) ACEMMEHSD17B10ALDH1A1SMN1; SMN2
SCHEMBL7342670 0.84 ACE (0.47) ACEMMEHSD17B10ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4808713-A Anthypertensive pyridazo [1,2-a][1,2]diazepines HOFFMAN-LA ROCHE INC. (US) 1989-02-28 US disclosed
US-4772701-A Pyridazo[1,2]pyridazines and pyrazolo[1,2]pyridazines as antihypertensives HOFFMANN-LA ROCHE INC. (US) 1988-09-20 US disclosed
US-4658024-A Pyrazolo [1,2-a][1,2]-diazepines useful as antihypertensives HOFFMANN-LA ROCHE INC. (US) 1987-04-14 US disclosed
US-4512924-A HYPOTENSIVE AGENTS HOFFMANN-LA ROCHE INC. (US) 1985-04-23 US disclosed
EP-0094095-A2 Bicyclic carboxylic acids and their alkyl and aralkyl esters F. HOFFMANN-LA ROCHE AG (CH) 1983-11-16 EP disclosed