SCHEMBL10567798

SCHEMBL10567798

CC(C)(C)C(=O)Nc1nc(O)c2c(n1)NCC(CNCc1ccc(C(=O)NC(CCC(=O)O)C(=O)O)c(Cl)c1)C2

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GART P22102 6/20 0.42
ATIC P31939 3/20 0.39
TYMS P04818 5/20 0.38
DHFR P00374 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10567793 1.00 GART (0.42) GARTATICTYMSDHFR
SCHEMBL9211571 0.89 GART (0.52) GARTATICTYMSDHFR
SCHEMBL10570448 0.89 GART (0.52) GARTATICTYMSDHFR
SCHEMBL9216949 0.88 GART (0.45) GARTATICTYMS
SCHEMBL9216933 0.88 GART (0.45) GARTATICTYMS
SCHEMBL10574310 0.83 GART (0.44) GARTATICTYMSDHFR
SCHEMBL10574300 0.83 GART (0.44) GARTATICTYMSDHFR
SCHEMBL9524154 0.80 GART (0.38) GARTDHFR
SCHEMBL9524143 0.80 GART (0.38) GARTDHFR
SCHEMBL10513249 0.78 TYMS (0.42) GARTATICTYMSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4871746-A N-[N-(tetrahydropyrido[2,3-D]pyrimidinylmethyl)-aminomethylbenzoyl]glutamic acid derivatives as neoplastic growth inhibitors THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-10-03 US disclosed