SCHEMBL9524154

SCHEMBL9524154

COC(=O)CC[C@@H](NC(=O)c1ccc(CCC2CNc3nc(NC(=O)C(C)(C)C)nc(O)c3C2)cc1Cl)C(=O)OC

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GART P22102 3/20 0.38
DHFR P00374 3/20 0.36
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524143 1.00 GART (0.38) GARTDHFRALDH1A1MAPK1
SCHEMBL10568483 0.88 GART (0.41) GARTDHFR
SCHEMBL9525469 0.88 GART (0.41) GARTDHFR
SCHEMBL9383820 0.86 DHFR (0.46) GARTDHFRALDH1A1MAPK1
SCHEMBL9383825 0.86 DHFR (0.46) GARTDHFRALDH1A1MAPK1
SCHEMBL8819377 0.85 GART (0.39) GARTDHFRALDH1A1
SCHEMBL8819374 0.85 GART (0.39) GARTDHFRALDH1A1
SCHEMBL9381115 0.84 GART (0.31) GART
SCHEMBL9381108 0.84 GART (0.31) GART
SCHEMBL9382961 0.83 DHFR (0.47) GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0327190-B1 Pyrido(2,3-d)pyrimidine derivatives UNIV PRINCETON (US) 1993-12-08 EP disclosed
US-4889859-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-12-26 US disclosed