SCHEMBL10567963

SCHEMBL10567963

CC(C(O)c1ccc(C(F)(F)F)cc1)n1cccn1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
CYP19A1 P11511 1/20 0.35
GPR139 Q6DWJ6 4/20 0.35
PDE2A O00408 2/20 0.35
PNMT P11086 1/20 0.34
ACP3 P15309 1/20 0.34
CASR P41180 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
TRPM8 Q7Z2W7 3/20 0.33
HSD11B1 P28845 1/20 0.33
CYP26A1 O43174 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP3A5 P20815 1/20 0.33
ALOX5AP P20292 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10566237 0.85 CYP19A1 (0.37) CYP19A1GPR139PDE2AACP3CASR
SCHEMBL10739867 0.82 GPR139 (0.40) GPR139PDE2A
SCHEMBL7091178 0.77 CYP19A1 (0.39) CES2CES1CYP19A1PDE2AACP3
SCHEMBL10360812 0.77 CYP3A4 (0.36) CYP19A1GPR139CASRCYP3A4CYP3A5
SCHEMBL10361513 0.76 CYP19A1 (0.42) CYP19A1CYP3A4ALOX5AP
SCHEMBL10568094 0.76 KCNH2 (0.37) CYP19A1GPR139PDE2ACASRCYP3A4
SCHEMBL10566838 0.74 CYP19A1 (0.37) CYP19A1CASRCYP3A4CYP3A5ALOX5AP
SCHEMBL10362527 0.73 GSK3B (0.46) CES2CES1CYP3A4
SCHEMBL10821169 0.71 CYP17A1 (0.41) CES2CES1CYP19A1PDE2A
SCHEMBL10568059 0.71 P2RX3 (0.43) CYP19A1CASRCYP3A4CYP3A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833159-A FUNGICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-23 US disclosed
US-4689337-A 1,2,4-TRIAZOLYL AND PYRAZOLYL GROUPS; FUNGICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-08-25 US disclosed
EP-0158448-A2 Azolyl propanols IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-10-16 EP disclosed