SCHEMBL10568204

SCHEMBL10568204

CCOC(=O)C1C(=O)Nc2cc3[nH]c(-c4nc[nH]n4)nc3cc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.39
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PKN1 Q16512 1/20 0.35
PKN2 Q16513 1/20 0.35
SIRT2 Q8IXJ6 6/20 0.35
SIRT1 Q96EB6 5/20 0.35
SIRT3 Q9NTG7 2/20 0.35
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
PDE3B Q13370 3/20 0.33
PDE3A Q14432 3/20 0.33
P2RY12 Q9H244 3/20 0.33
CHEK2 O96017 1/20 0.33
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32
HPSE Q9Y251 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10563558 0.82 TDP2 (0.41) TDP2ALDH1A1MAPTL3MBTL1PKN1
SCHEMBL9834430 0.82 TDP2 (0.45) TDP2ALDH1A1MAPTL3MBTL1KDM4E
SCHEMBL9833477 0.81 PKN1 (0.54) TDP2ALDH1A1MAPTL3MBTL1PKN1
SCHEMBL9833068 0.81 TDP2 (0.44) TDP2ALDH1A1MAPTL3MBTL1PKN1
SCHEMBL10566801 0.80 TDP2 (0.40) TDP2ALDH1A1MAPTL3MBTL1PKN1
SCHEMBL10566874 0.79 TDP2 (0.37) TDP2ALDH1A1MAPTL3MBTL1PKN1
SCHEMBL10567219 0.79 TDP2 (0.39) TDP2ALDH1A1MAPTL3MBTL1PKN1
SCHEMBL10567141 0.79 TDP2 (0.37) TDP2ALDH1A1MAPTL3MBTL1PKN1
SCHEMBL9833942 0.78 KDM4E (0.47) ALDH1A1MAPTPKN1PKN2KDM4E
SCHEMBL10571709 0.78 SIRT2 (0.39) TDP2ALDH1A1MAPTL3MBTL1PKN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed