SCHEMBL9833477

SCHEMBL9833477

CCOC(=O)C1C(=O)Nc2cc3[nH]c(-c4ccncc4)nc3cc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 2/20 0.54
PKN2 Q16513 2/20 0.54
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ALDH1A1 P00352 4/20 0.42
KDM4E B2RXH2 3/20 0.42
HPGD P15428 3/20 0.42
GAA P10253 1/20 0.42
SIRT2 Q8IXJ6 4/20 0.41
SIRT1 Q96EB6 3/20 0.41
SIRT3 Q9NTG7 1/20 0.41
TDP2 O95551 1/20 0.41
ALOX5 P09917 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9832273 0.89 PDE4A (0.48) PKN1PKN2PDE4APDE4BPDE4C
SCHEMBL9833942 0.89 KDM4E (0.47) PKN1PKN2NPC1RAB9AALDH1A1
SCHEMBL9830544 0.85 PDE4A (0.51) PKN1PKN2PDE4APDE4BPDE4C
SCHEMBL10571709 0.85 SIRT2 (0.39) PKN1PKN2NPC1RAB9AALDH1A1
SCHEMBL10563558 0.83 TDP2 (0.41) PKN1PKN2PDE3BPDE3ANPC1
SCHEMBL9834430 0.83 TDP2 (0.45) PDE3BPDE3ARAB9AALDH1A1KDM4E
SCHEMBL9833068 0.82 TDP2 (0.44) PKN1PKN2PDE3BPDE3AALDH1A1
SCHEMBL10567219 0.82 TDP2 (0.39) PKN1PKN2PDE3BPDE3ANPC1
SCHEMBL10566874 0.82 TDP2 (0.37) PKN1PKN2NPC1RAB9AALDH1A1
SCHEMBL10568204 0.81 TDP2 (0.39) PKN1PKN2PDE3BPDE3ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed