SCHEMBL10568243

SCHEMBL10568243

CC(C)=C1C(=O)Nc2cc3[nH]c(-c4ccnnc4)nc3cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
ALDH1A1 P00352 5/20 0.36
HPGD P15428 4/20 0.36
KDM4E B2RXH2 4/20 0.36
GAA P10253 1/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
STAT1 P42224 1/20 0.36
MITF O75030 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
BRD4 O60885 7/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831955 0.87 PDE3B (0.53) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9831891 0.86 MAPT (0.54) ALDH1A1HPGDKDM4EHSD17B10NPC1
SCHEMBL9836597 0.76 EGFR (0.36) BRD4
SCHEMBL9834857 0.76 HSP90AA1 (0.39) ALDH1A1HPGDKDM4ERAB9AMAPT
SCHEMBL10567700 0.75 BRD4 (0.33) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10566025 0.74 PDE3B (0.69) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10373348 0.73 CDK4 (0.40) PDE3BPDE3ABRD4
SCHEMBL10567302 0.73 PDE3B (0.41) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10569319 0.71 PDE4A (0.40) PDE4APDE4BPDE4CPDE4DPDE3B
Hydrochloric Acid SCHEMBL10560128 0.69 PDE4A (0.42) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed