SCHEMBL10567302

SCHEMBL10567302

CC1C(=O)Nc2cc3[nH]c(-c4ccnnc4)nc3cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
ALDH1A1 P00352 5/20 0.37
HPGD P15428 5/20 0.37
KDM4E B2RXH2 4/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
MAPT P10636 2/20 0.37
STAT1 P42224 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10470299 0.87 PDE3B (0.55) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10569319 0.86 PDE4A (0.40) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10477754 0.83 NPBWR1 (0.46) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10567486 0.80 PDE4A (0.35) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10477810 0.79 TCF4 (0.51) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10567103 0.78 PGR (0.37) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10373856 0.76 FBP1 (0.55) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10569181 0.75 NPC1 (0.43) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10566025 0.75 PDE3B (0.69) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10566128 0.75 PDE3B (0.34) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed