SCHEMBL9834857

SCHEMBL9834857

CC(C)=C1C(=O)Nc2cc3[nH]c(C)nc3cc21

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.39
ESR2 Q92731 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HPGD P15428 3/20 0.37
POLB P06746 2/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 3/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
BRD4 O60885 11/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
BRD2 P25440 1/20 0.34
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836597 0.86 EGFR (0.36) BRD4BRD2EGFR
SCHEMBL9831955 0.78 PDE3B (0.53) HPGDPOLBMAPTKDM4EALDH1A1
SCHEMBL10567700 0.77 BRD4 (0.33) RAB9ABRD4BRD2
SCHEMBL10568243 0.76 PDE4A (0.40) HPGDPOLBMAPTKDM4EALDH1A1
SCHEMBL9831891 0.75 MAPT (0.54) HPGDPOLBMAPTKDM4EALDH1A1
SCHEMBL10373348 0.73 CDK4 (0.40) BRD4BRD2EGFR
SCHEMBL13041691 0.68 ALDH1A1 (0.59) HSP90AA1ESR2TDP1HPGDPOLB
SCHEMBL20436361 0.67 BRD4 (0.57) MAPTKDM4EALDH1A1BRD4BRD2
SCHEMBL8135807 0.67 HPGD (0.44) HSP90AA1ESR2TDP1HPGDPOLB
SCHEMBL9835803 0.67 HSP90AA1 (0.40) HSP90AA1ESR2TDP1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214592-B1 PYRROLOBENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE PRODUCTS Roche Diagnostics GmbH (DE) 1991-08-14 EP disclosed
US-4730003-A Tricyclic compounds for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-03-08 US disclosed
EP-0214592-A2 Pyrrolobenzimidazoles, process for their preparation and medicaments containing these products Roche Diagnostics GmbH (DE) 1987-03-18 EP disclosed