SCHEMBL10568269

SCHEMBL10568269

CON1C(=O)CC2(CCN(C(C)=O)CC2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.36
CHRM3 P20309 1/20 0.36
USP2 O75604 2/20 0.35
CYP2D6 P10635 4/20 0.34
ALDH1A1 P00352 3/20 0.34
CYP2C19 P33261 3/20 0.34
TSHR P16473 2/20 0.34
MAPK1 P28482 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CYP2C9 P11712 4/20 0.33
GAA P10253 1/20 0.33
GFER P55789 1/20 0.33
CYP3A4 P08684 3/20 0.33
CYP1A2 P05177 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
MMP3 P08254 1/20 0.32
MMP10 P09238 1/20 0.32
LMNA P02545 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10565385 0.84 POLB (0.42) CHRM2CHRM3CYP2D6ALDH1A1CYP2C19
Hydrochloric Acid SCHEMBL10565807 0.81 ITGB3 (0.37) CHRM2CHRM3ALDH1A1MEN1KMT2A
SCHEMBL10568268 0.81 USP30 (0.42) USP2TSHRTHRBHPGD
SCHEMBL10563612 0.78 KCNH2 (0.33) CHRM2CHRM3ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL10563363 0.72 CHRM2 (0.33) CHRM2CHRM3
SCHEMBL18711765 0.71 USP2 (0.41) USP2CYP2D6ALDH1A1CYP2C19TSHR
SCHEMBL27256625 0.69 CYP1A2 (0.43) USP2CYP2D6ALDH1A1CYP2C19TSHR
Hydrochloric Acid SCHEMBL10563441 0.69 CHRM2 (0.30) CHRM2CHRM3ALDH1A1HPGD
SCHEMBL18711770 0.68 USP2 (0.39) USP2CYP2D6ALDH1A1CYP2C19TSHR
SCHEMBL18711764 0.67 USP2 (0.38) USP2CYP2D6ALDH1A1CYP2C19TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4804665-A NERVOUS SYSTEM DISORDERS; COGNITION ACTIVATORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1989-02-14 US disclosed
EP-0273659-A1 Azaspiro compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1988-07-06 EP disclosed