Closiramine

Closiramine

SCHEMBL10568448

CN(C)CCC1c2ccc(Cl)cc2CCc2cccnc21

nearest known ligand 0.75

Full drug profile on Sugi Atlas →

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.75
KMT2A Q03164 1/20 0.75
ATM Q13315 1/20 0.75
FNTA P49354 10/20 0.50
FNTB P49356 10/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Closiramine SCHEMBL637355 0.87 MEN1 (1.00) MEN1KMT2AATMFNTAFNTB
SCHEMBL14102189 0.86 MEN1 (0.58) MEN1KMT2AATMFNTAFNTB
SCHEMBL14288461 0.84 MEN1 (0.56) MEN1KMT2AATMFNTAFNTB
SCHEMBL14102072 0.84 MEN1 (0.58) MEN1KMT2AATMFNTAFNTB
SCHEMBL14102079 0.84 MEN1 (0.56) MEN1KMT2AATMFNTAFNTB
SCHEMBL14102196 0.80 MEN1 (0.53) MEN1KMT2AATMFNTAFNTB
SCHEMBL14101997 0.77 MEN1 (0.50) MEN1KMT2AATMFNTAFNTB
SCHEMBL13611706 0.77 FNTA (0.58) MEN1KMT2AATMFNTAFNTB
SCHEMBL14102242 0.76 MEN1 (0.49) MEN1KMT2AATMFNTAFNTB
SCHEMBL1978262 0.75 FNTA (0.60) FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114748624-A Composition for treating or preventing vasomotor symptoms 田边三菱制药株式会社 2022-07-15 CN disclosed
US-20220047505-A1 Controlled Absorption Water-Soluble Pharmaceutically Active Organic Compound Formulation for Once-Daily Administration STI PHARMA, LLC (US) 2022-02-17 US disclosed
US-4831042-A Tricyclic-substituted piperidine antihistamines SCHERING CORPORATION (US) 1989-05-16 US disclosed
US-4560688-A NON-SEDATING; CARBAMOYL OR SULFONAMIDE DERIVATIVES SCHERING CORPORATION (US) 1985-12-24 US disclosed
US-4454143-A Tricyclic antihistamines SCHERING CORPORATION (US) 1984-06-12 US disclosed
US-4355036-A Tricyclic-substituted piperidine antihistamines SCHERING CORPORATION (US) 1982-10-19 US disclosed