SCHEMBL10568502

SCHEMBL10568502

CCC1(CC)C(=O)Nc2cc3[nH]c(-c4ccco4)nc3cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.47
EPHX2 P34913 1/20 0.47
ALDH1A1 P00352 5/20 0.46
RAB9A P51151 4/20 0.46
KDM4E B2RXH2 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
CHEK1 O14757 1/20 0.46
LIMK1 P53667 1/20 0.46
CDK5 Q00535 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
MAPT P10636 4/20 0.45
POLB P06746 3/20 0.45
HSD17B10 Q99714 3/20 0.45
KMT2A Q03164 2/20 0.45
PKM P14618 1/20 0.45
NPC1 O15118 3/20 0.42
TP53 P04637 3/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10567229 0.85 PDE4A (0.56) ALOX5EPHX2ALDH1A1RAB9AKDM4E
SCHEMBL10373500 0.81 PDE4A (0.51) ALDH1A1RAB9AKDM4ESMN1; SMN2MAPT
SCHEMBL9832933 0.78 PDE4A (0.65) ALDH1A1RAB9AKDM4EMAPTHSD17B10
SCHEMBL9832117 0.77 MAPT (0.54) EPHX2ALDH1A1RAB9AKDM4ESMN1; SMN2
SCHEMBL9833966 0.76 MAPT (0.40) ALDH1A1RAB9AKDM4ESMN1; SMN2MAPT
SCHEMBL10530446 0.74 CHEK1 (0.49) ALOX5EPHX2ALDH1A1RAB9AKDM4E
SCHEMBL10698980 0.73 AURKA (0.57) ALOX5EPHX2ALDH1A1RAB9AKDM4E
SCHEMBL10566214 0.73 ALOX5 (0.52) ALOX5EPHX2ALDH1A1RAB9AKDM4E
SCHEMBL10373365 0.72 PDE2A (0.45) ALDH1A1RAB9AKDM4ESMN1; SMN2MAPT
SCHEMBL10699765 0.72 AURKA (0.48) ALOX5EPHX2ALDH1A1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed