SCHEMBL10568720

SCHEMBL10568720

CN1C(=O)CCc2c1ccc(OCCN1CCN(c3ccccc3)CC1)c2Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.48
DRD2 P14416 7/20 0.47
DRD3 P35462 5/20 0.47
DRD1 P21728 1/20 0.47
DRD5 P21918 1/20 0.47
DRD4 P21917 2/20 0.43
ADRB2 P07550 1/20 0.43
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
ADRB1 P08588 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
SIGMAR1 Q99720 2/20 0.42
HTR2A P28223 1/20 0.42
HRH1 P35367 1/20 0.42
TMEM97 Q5BJF2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10572119 0.86 HTR1A (0.57) HTR1ADRD2DRD3DRD1DRD5
SCHEMBL10572762 0.84 MAPT (0.51)
SCHEMBL10570087 0.82 HTR1A (0.47) HTR1ADRD2DRD3DRD1DRD5
SCHEMBL10570155 0.81 HTR1A (0.57) HTR1ADRD2DRD3DRD4ADRB2
SCHEMBL11064799 0.77 TMEM97 (0.53) DRD2DRD3DRD4ADRB2CHRM2
SCHEMBL10575317 0.72 SIGMAR1 (0.54) HTR1ADRD2DRD3DRD1DRD5
SCHEMBL10569223 0.72 SIGMAR1 (0.56) HTR1ADRD2DRD3DRD1DRD5
SCHEMBL10573223 0.72 DRD3 (0.60) HTR1ADRD2DRD3ADRA1ASIGMAR1
SCHEMBL10569856 0.71 MAPT (0.59) ADRB2ADRB1
Hydrochloric Acid SCHEMBL10668121 0.70 MAPT (0.59)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4824840-A ANTIHISTAMINES, NERVOUS SYSTEM CONTROLLERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-04-25 US disclosed
US-4734416-A ANTIHISTAMINES, CENTRAL NERVOUS SYSTEM CONTROLLING ACTION OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-03-29 US disclosed