SCHEMBL10569263

SCHEMBL10569263

CCOC(=O)C1(C)C(=O)Nc2cc3c(cc21)NC(c1ccncn1)N3

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.32
LMNA P02545 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PDE5A O76074 1/20 0.32
ADCY8 P40145 1/20 0.32
FGB P02675 1/20 0.31
NAMPT P43490 1/20 0.31
MAPT P10636 1/20 0.31
KDM4E B2RXH2 1/20 0.30
CASP1 P29466 1/20 0.30
HSD17B10 Q99714 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10566881 0.86 MAPT (0.32) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL9831490 0.85 KDM4E (0.37) BRD4ALDH1A1TP53CYP1A2CYP3A4
SCHEMBL10569723 0.85 MAPT (0.31) ALDH1A1TP53CYP1A2CYP3A4CYP2C9
SCHEMBL10567540 0.85 PDE5A (0.32) BRD4LMNAALDH1A1TP53CYP1A2
Hydrochloric Acid SCHEMBL10470525 0.85 KDM4E (0.36) BRD4ALDH1A1TP53CYP1A2CYP3A4
SCHEMBL10566715 0.84 KDM5A (0.31)
SCHEMBL10568374 0.82 BRD4 (0.34) BRD4LMNAALDH1A1TP53CYP1A2
SCHEMBL9833624 0.80 KDM4E (0.46) ALDH1A1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL10567876 0.79 PDE3B (0.42)
SCHEMBL9835044 0.79 SMN1; SMN2 (0.41) BRD4LMNAALDH1A1TP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed