SCHEMBL10569723

SCHEMBL10569723

CCOC(=O)C1(C)C(=O)Nc2cc3c(cc21)NC(c1cnncn1)N3

nearest known ligand 0.31

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.31
PDE5A O76074 1/20 0.31
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
ADCY8 P40145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10566881 0.87 MAPT (0.32) MAPTALDH1A1TP53CYP1A2CYP3A4
SCHEMBL10567540 0.86 PDE5A (0.32) MAPTPDE5AALDH1A1TP53CYP1A2
SCHEMBL10569263 0.85 BRD4 (0.32) MAPTPDE5AALDH1A1TP53CYP1A2
SCHEMBL10569956 0.81 ALDH1A1 (0.33) MAPTPDE5AALDH1A1TP53CYP1A2
SCHEMBL10568374 0.81 BRD4 (0.34) MAPTPDE5AALDH1A1TP53CYP1A2
SCHEMBL10567457 0.79 ADORA2B (0.33) MAPTALDH1A1TP53CYP1A2CYP3A4
SCHEMBL9833652 0.79 ALDH1A1 (0.36) MAPTALDH1A1TP53CYP1A2CYP3A4
SCHEMBL10569268 0.78 PDE5A (0.32) PDE5A
SCHEMBL9831490 0.78 KDM4E (0.37) MAPTALDH1A1TP53CYP1A2CYP3A4
SCHEMBL9835788 0.78 MAPT (0.36) MAPTALDH1A1TP53CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed