SCHEMBL10568374

SCHEMBL10568374

CCOC(=O)C1(C)C(=O)Nc2cc3c(cc21)NC(c1cccnn1)N3

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
ADCY8 P40145 1/20 0.33
PDE5A O76074 1/20 0.33
FGB P02675 1/20 0.33
KDM4E B2RXH2 4/20 0.32
CASP1 P29466 2/20 0.32
HSD17B10 Q99714 1/20 0.32
LMNA P02545 1/20 0.32
ALDH1A1 P00352 4/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32
KCNH2 Q12809 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10569263 0.82 BRD4 (0.32) BRD4ADCY8PDE5AFGBKDM4E
SCHEMBL9833624 0.82 KDM4E (0.46) KDM4ECASP1HSD17B10ALDH1A1SMN1; SMN2
SCHEMBL9831490 0.81 KDM4E (0.37) BRD4ADCY8FGBKDM4ECASP1
SCHEMBL9835044 0.81 SMN1; SMN2 (0.41) BRD4ADCY8KDM4ELMNAALDH1A1
SCHEMBL10569723 0.81 MAPT (0.31) ADCY8PDE5AALDH1A1SMN1; SMN2TP53
SCHEMBL10567540 0.81 PDE5A (0.32) BRD4ADCY8PDE5AKDM4ECASP1
Hydrochloric Acid SCHEMBL10470525 0.81 KDM4E (0.36) BRD4ADCY8FGBKDM4ECASP1
SCHEMBL10566881 0.80 MAPT (0.32) ADCY8FGBALDH1A1SMN1; SMN2TP53
SCHEMBL10566478 0.79 PDE3B (0.40)
SCHEMBL9833693 0.79 ALDH1A1 (0.36) BRD4ADCY8PDE5AFGBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4835280-A Indoline compounds for synthesis of pharmaceutically active pyrrolobenzimidazoles BOEHRINGER MANNHEIM GMBH (DE) 1989-05-30 US disclosed
US-4695567-A Pyrrolobenzimidazoles, pharmaceutical compositions containing them and method of using them to treat certain heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1987-09-22 US disclosed
EP-0189103-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1986-07-30 EP disclosed