SCHEMBL10572425

SCHEMBL10572425

CCC(Oc1cccc2c1CCC(=O)N2)N1CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.43
OPRK1 P41145 2/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
SCN1A P35498 2/20 0.35
SCN5A Q14524 2/20 0.35
SCN9A Q15858 2/20 0.35
SLC6A2 P23975 5/20 0.34
SLC6A4 P31645 5/20 0.34
KCNH2 Q12809 4/20 0.34
CYP3A4 P08684 4/20 0.34
CYP2D6 P10635 4/20 0.34
CACNA1F O60840 2/20 0.34
CACNA1D Q01668 2/20 0.34
CACNA1S Q13698 2/20 0.34
CACNA1C Q13936 2/20 0.34
SLC6A3 Q01959 1/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
CHRM2 P08172 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11282871 0.74 ADRB1 (0.49) HTR1AOPRK1ADRB2ADRB1SCN1A
SCHEMBL10573123 0.73 ADRB2 (0.44) HTR1AOPRK1ADRB2ADRB1SCN1A
SCHEMBL10572437 0.72 HRH3 (0.49) HTR1AOPRK1ADRB2ADRB1DRD2
SCHEMBL11285594 0.72 ADRB1 (0.47) HTR1AOPRK1ADRB2ADRB1SCN1A
SCHEMBL1764193 0.72 ADRB2 (0.57) HTR1AOPRK1ADRB2ADRB1DRD2
SCHEMBL9653563 0.72 ADRB1 (0.49) HTR1AOPRK1ADRB2ADRB1SCN1A
SCHEMBL11539715 0.71 HTR2C (0.46) HTR1AADRB1SLC6A2SLC6A4KCNH2
SCHEMBL11283090 0.71 ADRB2 (0.48) HTR1AOPRK1ADRB2ADRB1KDM4E
SCHEMBL27691792 0.70 ADRB1 (0.53) HTR1AOPRK1ADRB2ADRB1SCN1A
SCHEMBL30636067 0.70 ADRB2 (0.51) HTR1AOPRK1ADRB2ADRB1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4824840-A ANTIHISTAMINES, NERVOUS SYSTEM CONTROLLERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1989-04-25 US disclosed