SCHEMBL10600285

SCHEMBL10600285

C=CC(N)n1cnc2c(=O)n(C)c(=O)n(C)c21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.45
ALDH1A1 P00352 4/20 0.38
HTT P42858 2/20 0.38
POLB P06746 2/20 0.36
ADORA2B P29275 5/20 0.36
MAPT P10636 2/20 0.35
HSD17B10 Q99714 1/20 0.34
TP53 P04637 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ADORA2A P29274 3/20 0.33
PIK3CD O00329 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CNR1 P21554 1/20 0.33
ACHE P22303 1/20 0.33
ADORA1 P30542 1/20 0.33
NTSR1 P30989 1/20 0.33
MC3R P41968 1/20 0.33
NOTUM Q6P988 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17682185 0.77 LMNA (0.50) LMNAALDH1A1HTTPOLBADORA2B
SCHEMBL19601295 0.76 LMNA (0.49) LMNAALDH1A1HTTPOLBADORA2B
SCHEMBL11190463 0.75 LMNA (0.46) LMNAALDH1A1HTTPOLBADORA2B
SCHEMBL23974577 0.74 LMNA (0.54) LMNAALDH1A1HTTPOLBADORA2B
SCHEMBL3272841 0.72 LMNA (0.54) LMNAALDH1A1HTTPOLBADORA2B
Isocaffiene SCHEMBL515995 0.71 LMNA (0.57) LMNAALDH1A1HTTPOLBADORA2B
SCHEMBL1962417 0.70 LMNA (0.69) LMNAALDH1A1HTTPOLBADORA2B
SCHEMBL8136340 0.68 LMNA (0.54) LMNAALDH1A1HTTPOLBADORA2B
SCHEMBL28048679 0.68 LMNA (0.54) LMNAALDH1A1HTTPOLBADORA2B
SCHEMBL11187813 0.67 LMNA (0.52) LMNAALDH1A1HTTPOLBADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0077896-B1 THEOPHYLLINE DERIVATIVES, ANTIBODIES AND THEIR PREPARATION FROM THEOPHYLLINE IMMUNOGENS, AS WELL AS AN IMMUNO ASSAY METHOD AND REAGENT MEANS FOR DETERMINING THEOPHYLLINE MILES INC. (US) 1989-01-25 EP disclosed
US-4608336-A DETERMINATION OF THEOPHYLLINE IN BIOLOGICAL FLUIDS MILES LABORATORIES, INC. (US) 1986-08-26 US disclosed
US-4533493-A IMMUNOASSAYS FOR MEASUREMENT OF THEOPHYLLINE IN BIOLOGIACAL FLUIDS MILES LABORATORIES, INC. (US) 1985-08-06 US disclosed
US-4460772-A IMMUNOASSAY MILES LABORATORIES, INC. (US) 1984-07-17 US disclosed
EP-0077896-A1 Theophylline derivatives, antibodies and their preparation from theophylline immunogens, as well as an immuno assay method and reagent means for determining theophylline MILES INC. (US) 1983-05-04 EP disclosed