SCHEMBL10604647

SCHEMBL10604647

O=C1c2ccccc2OC(CCCCCO)c2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.39
STK17B O94768 1/20 0.37
ADORA3 P0DMS8 1/20 0.36
AR P10275 1/20 0.36
HSD11B1 P28845 1/20 0.36
AKR1C3 P42330 1/20 0.36
PKM P14618 1/20 0.36
TSHR P16473 1/20 0.36
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4021498 0.84 ALDH1A1 (0.47) CES2
SCHEMBL9870428 0.84 EDNRB (0.40) EDNRBEDNRA
SCHEMBL27667860 0.82 ALDH1A1 (0.48)
SCHEMBL19283540 0.77 ALDH1A1 (0.49)
SCHEMBL29756436 0.77 ALDH1A1 (0.49)
SCHEMBL2728660 0.71 ALDH1A1 (0.51)
SCHEMBL7599711 0.70 ABCB1 (0.48) ADORA3ARHSD11B1AKR1C3
SCHEMBL7872301 0.69 CES2 (0.61) CES2
SCHEMBL7876620 0.69 CES2 (0.61) CES2
SCHEMBL1463773 0.69 CES2 (0.61) CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0160258-B1 (6,11-DIHYDRO-11-OXODIBENZ(BM,E)OXEPINYL)PENTANOLS, A PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-09-27 EP disclosed
EP-0160258-B1 (6,11-DIHYDRO-11-OXODIBENZ(BM,E)OXEPINYL)PENTANOLS, A PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-09-27 EP disclosed
EP-0160258-A2 (6,11-Dihydro-11-oxodibenz(bm,e)oxepinyl)pentanols, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1985-11-06 EP disclosed
EP-0160258-A2 (6,11-Dihydro-11-oxodibenz(bm,e)oxepinyl)pentanols, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1985-11-06 EP disclosed