SCHEMBL10606244

SCHEMBL10606244

COc1ccccc1OC1CCN(C(=O)Cl)C1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.56
PDE4B Q07343 11/20 0.46
PDE10A Q9Y233 1/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
PDE4A P27815 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10608977 0.86 EPHX2 (0.56) EPHX2PDE10AMEN1KMT2A
SCHEMBL10606038 0.86 EPHX2 (0.50) EPHX2PDE4BPDE10APDE4APDE4C
SCHEMBL10608868 0.85 DGAT2 (0.53)
SCHEMBL23365281 0.81 EPHX2 (0.62) EPHX2PDE4BMEN1KMT2A
SCHEMBL14413529 0.81 EPHX2 (0.59) EPHX2PDE4BMEN1KMT2APDE4A
SCHEMBL10609876 0.81 HCRTR1 (0.48) EPHX2PDE10AMEN1KMT2A
SCHEMBL10605998 0.80 EPHX2 (0.53) EPHX2KMT2A
SCHEMBL10606119 0.80 EPHX2 (0.54) EPHX2
SCHEMBL10608410 0.80 EPHX2 (0.46) EPHX2
SCHEMBL10605809 0.78 EPHX2 (0.56) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0147909-B1 ARYLOXY-N-(AMINOALKYL)-1-PYRROLIDINE AND PIPERIDINE CARBOXAMIDES AND CARBOTHIOAMIDES HAVING ANTIARRHYTHMIC ACTIVITY A.H. ROBINS COMPANY, INCORPORATED (US) 1989-12-06 EP disclosed
US-4547514-A Aryloxy-N-(aminoalkyl)-1-pyrrolidine and piperidine carboxamides and carbothioamides having antiarrhythmic activity A. H. ROBINS COMPANY, INCORPORATED (US) 1985-10-15 US disclosed
EP-0147909-A1 Aryloxy-N-(aminoalkyl)-1-pyrrolidine and piperidine carboxamides and carbothioamides having antiarrhythmic activity A.H. ROBINS COMPANY, INCORPORATED (US) 1985-07-10 EP disclosed