SCHEMBL10608977

SCHEMBL10608977

Cc1ccccc1OC1CCN(C(=O)Cl)C1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.56
KMT2A Q03164 3/20 0.52
SCD O00767 1/20 0.46
HRH3 Q9Y5N1 1/20 0.45
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
PDE10A Q9Y233 1/20 0.42
HRH1 P35367 2/20 0.42
KDM4E B2RXH2 1/20 0.41
NPY1R P25929 1/20 0.41
NPY2R P49146 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 1/20 0.41
BCAT2 O15382 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28278842 0.87 EPHX2 (0.57) EPHX2KMT2ASCDHRH3NPC1
SCHEMBL10609005 0.86 EPHX2 (0.50) EPHX2KMT2ASCDHRH3NPC1
SCHEMBL10606244 0.86 EPHX2 (0.56) EPHX2KMT2APDE10AMEN1
SCHEMBL10608868 0.83 DGAT2 (0.53)
SCHEMBL9903544 0.81 EPHX2 (0.62) EPHX2KMT2ASCDHRH3NPC1
SCHEMBL15061997 0.81 EPHX2 (0.59) EPHX2KMT2ASCDNPC1RAB9A
SCHEMBL10609876 0.81 HCRTR1 (0.48) EPHX2KMT2ARAB9APDE10AKDM4E
SCHEMBL10606119 0.80 EPHX2 (0.54) EPHX2
SCHEMBL10608410 0.80 EPHX2 (0.46) EPHX2SCDHRH1KDM4E
SCHEMBL10610446 0.78 SSTR4 (0.43) EPHX2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0147909-B1 ARYLOXY-N-(AMINOALKYL)-1-PYRROLIDINE AND PIPERIDINE CARBOXAMIDES AND CARBOTHIOAMIDES HAVING ANTIARRHYTHMIC ACTIVITY A.H. ROBINS COMPANY, INCORPORATED (US) 1989-12-06 EP disclosed
US-4547514-A Aryloxy-N-(aminoalkyl)-1-pyrrolidine and piperidine carboxamides and carbothioamides having antiarrhythmic activity A. H. ROBINS COMPANY, INCORPORATED (US) 1985-10-15 US disclosed
EP-0147909-A1 Aryloxy-N-(aminoalkyl)-1-pyrrolidine and piperidine carboxamides and carbothioamides having antiarrhythmic activity A.H. ROBINS COMPANY, INCORPORATED (US) 1985-07-10 EP disclosed