SCHEMBL10608205

SCHEMBL10608205

Cc1[nH]c(=O)sc1C(=O)c1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 2/20 0.48
CCNA2 P20248 8/20 0.46
CDK2 P24941 8/20 0.46
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
MAP2K1 Q02750 1/20 0.44
ALDH1A1 P00352 2/20 0.44
APP P05067 1/20 0.44
GAA P10253 1/20 0.44
HCAR3 P49019 1/20 0.44
HCAR2 Q8TDS4 1/20 0.44
F7 P08709 1/20 0.42
F3 P13726 1/20 0.42
SARM1 Q6SZW1 1/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
SIRT6 Q8N6T7 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
SIRT3 Q9NTG7 1/20 0.42
SIRT5 Q9NXA8 1/20 0.42
SIRT4 Q9Y6E7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10608201 0.82 CCNA2 (0.44) CHRM4CCNA2CDK2CDK5CDK5R1
SCHEMBL10605822 0.82 CHRM4 (0.44) CHRM4CCNA2CDK2KMT2A
SCHEMBL10628206 0.82 ALDH1A1 (0.43) CHRM4CCNA2CDK2ALDH1A1KMT2A
SCHEMBL9484144 0.72 MAP2K1 (0.48) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL29915528 0.72 ALDH1A1 (0.71) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL1242243 0.72 ALDH1A1 (0.71) MAP2K1ALDH1A1APPGAAHCAR3
SCHEMBL10662778 0.71 CHRM4 (0.57) CHRM4CCNA2CDK2CDK5CDK5R1
SCHEMBL10473732 0.71 MEN1 (0.53) CCNA2CDK2ALDH1A1GAAKMT2A
SCHEMBL10628308 0.71 ESR1 (0.44) ALDH1A1GAAKMT2A
Hydrochloric Acid SCHEMBL27841975 0.70 ALDH1A1 (0.68) MAP2K1ALDH1A1APPGAAHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1020730-C PREPARING METHOD FOR THIAZOLKETONE ADDITIVE MERRELL DOW PHARMA (US) 1993-05-19 CN disclosed
EP-0219625-B1 CARDIOTONIC HETEROCYCLOCARBONYL- AND ACETYL-THIAZOLONES MERRELL DOW PHARMACEUTICALS INC. (US) 1989-11-29 EP disclosed
EP-0219625-A1 Cardiotonic heterocyclocarbonyl- and acetyl-thiazolones MERRELL DOW PHARMACEUTICALS INC. (US) 1987-04-29 EP disclosed
CN-86104968-A Cardiotonic heterocyclic carbonyl and acetyl thiazolones 1987-04-22 CN disclosed
US-4623651-A Cardiotonic heterocyclocarbonyl- and acetyl-thiazolones MERRELL DOW PHARMACEUTICALS INC. (US) 1986-11-18 US disclosed