SCHEMBL10638166

SCHEMBL10638166

Cc1cnn(-c2nc3ccccc3c(=O)[nH]2)c1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.61
TNKS2 Q9H2K2 4/20 0.53
PARP1 P09874 3/20 0.53
HTR3A P46098 1/20 0.52
EGLN1 Q9GZT9 3/20 0.52
TNKS O95271 2/20 0.49
SPR P35270 3/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
QTRT1 Q9BXR0 1/20 0.45
KDM4E B2RXH2 3/20 0.45
KMT2A Q03164 2/20 0.45
CASP3 P42574 1/20 0.45
SENP8 Q96LD8 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10633932 0.83 GUSB (0.49) MGLLTNKS2PARP1HTR3AEGLN1
SCHEMBL10637521 0.83 TNKS2 (0.52) MGLLTNKS2PARP1HTR3AEGLN1
SCHEMBL10640119 0.83 NPC1 (0.52) MGLLTNKS2PARP1HTR3AEGLN1
SCHEMBL10634743 0.82 HTR3A (0.56) MGLLTNKS2PARP1HTR3AEGLN1
SCHEMBL10640495 0.82 EGLN1 (0.51) MGLLTNKS2PARP1HTR3AEGLN1
SCHEMBL10638059 0.82 EGLN1 (0.51) MGLLHTR3AEGLN1KMT2ACASP3
SCHEMBL10638241 0.81 PARP1 (0.55) MGLLTNKS2PARP1EGLN1TNKS
SCHEMBL3025892 0.81 EGLN1 (0.72) EGLN1
SCHEMBL10640188 0.80 MGLL (0.48) MGLLTNKS2PARP1HTR3AEGLN1
SCHEMBL10633927 0.79 EGLN1 (0.54) MGLLEGLN1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4644000-A FUNGICIDES, BACTERICIDES, SLIMICIDES BAYER AKTIENGESELLSCHAFT (DE) 1987-02-17 US claimed
EP-0161418-B1 ANTIMICROBIAL AGENTS CONTAINING 2-(1H-PYRAZOL-1-YL)-4-(3H)-QUINAZOLINONES BAYER AG (DE) 1988-09-07 EP disclosed
US-4644000-A FUNGICIDES, BACTERICIDES, SLIMICIDES BAYER AKTIENGESELLSCHAFT (DE) 1987-02-17 US disclosed
EP-0161418-A1 Antimicrobial agents containing 2-(1H-pyrazol-1-yl)-4-(3H)-quinazolinones BAYER AG (DE) 1985-11-21 EP disclosed