SCHEMBL10642181

SCHEMBL10642181

CCN(CC)CCCCC1CCCCN1CCNC(=O)N1c2ccccc2CC(=O)c2csc(C)c21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.42
CHRM4 P08173 3/20 0.42
CHRM1 P11229 3/20 0.42
CHRM3 P20309 3/20 0.42
CYP1A2 P05177 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MEN1 O00255 1/20 0.42
ALOX15 P16050 1/20 0.42
KMT2A Q03164 1/20 0.42
CHRM5 P08912 1/20 0.42
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TP53 P04637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824875 0.87 CHRM2 (0.56) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10647108 0.85 HRH3 (0.41) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10643569 0.77 BCHE (0.44) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL9824001 0.77 CHRM2 (0.63) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10644480 0.74 CHRM2 (0.58) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL9824650 0.72 CHRM2 (0.78) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL9824376 0.71 CYP1A2 (0.54) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10642067 0.71 CHRM2 (0.67) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL10641736 0.71 CHRM2 (0.75) CHRM2CHRM4CHRM1CHRM3CYP1A2
SCHEMBL9824697 0.70 CHRM2 (0.57) CHRM2CHRM4CHRM1CHRM3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273239-A1 Condensed diazepinones, processes for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1988-07-06 EP disclosed