SCHEMBL9824875

SCHEMBL9824875

CCN(CC)CCCCC1CCCCN1CCNC(=O)N1c2ccccc2NC(=O)c2csc(C)c21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 6/20 0.56
CHRM1 P11229 5/20 0.52
CHRM3 P20309 5/20 0.52
CHRM4 P08173 4/20 0.52
CYP1A2 P05177 3/20 0.52
CYP3A4 P08684 3/20 0.52
CYP2D6 P10635 2/20 0.52
CYP2C9 P11712 2/20 0.52
CYP2C19 P33261 2/20 0.52
ALOX15 P16050 2/20 0.52
CHRM5 P08912 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.41
DRD1 P21728 1/20 0.41
DRD5 P21918 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9824001 0.91 CHRM2 (0.63) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL10642181 0.87 CHRM2 (0.42) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL9824376 0.85 CYP1A2 (0.54) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL9824697 0.84 CHRM2 (0.57) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL9824056 0.83 CHRM2 (0.62) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL9824650 0.81 CHRM2 (0.78) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL9824863 0.80 CHRM2 (0.51) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL9824022 0.79 CHRM2 (0.79) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL9824296 0.78 ALDH1A1 (0.53) CHRM2CHRM1CHRM3CHRM4CYP1A2
SCHEMBL9824476 0.78 CHRM2 (0.59) CHRM2CHRM1CHRM3CHRM4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273239-B1 CONDENSED DIAZEPINONES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1991-03-06 EP disclosed
EP-0273239-A1 Condensed diazepinones, processes for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1988-07-06 EP disclosed