SCHEMBL1064228

SCHEMBL1064228

C[C@@H](c1ccc(C(=O)O)cc1)n1c(=O)[nH]c2ccccc2c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.48
ALDH1A1 P00352 4/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
KDM4E B2RXH2 3/20 0.47
HPGD P15428 2/20 0.47
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
CA12 O43570 1/20 0.46
RNASEH1 O60930 1/20 0.46
ERCC1 P07992 1/20 0.46
ERCC5 P28715 1/20 0.46
FEN1 P39748 1/20 0.46
CA9 Q16790 1/20 0.46
ERCC4 Q92889 1/20 0.46
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
B3GNT2 Q9NY97 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1064229 1.00 MAPK1 (0.48) MAPK1ALDH1A1L3MBTL1KDM4EHPGD
SCHEMBL1058359 0.86 KIF11 (0.49) MAPK1ALDH1A1L3MBTL1KDM4EHPGD
SCHEMBL6215191 0.83 MAPK1 (0.46) MAPK1KMT2AMEN1B3GNT2POLB
SCHEMBL6216031 0.83 B3GNT2 (0.46) MAPK1ALDH1A1KDM4EHPGDCA12
SCHEMBL3685482 0.83 ALDH1A1 (0.51) MAPK1ALDH1A1L3MBTL1KDM4EHPGD
SCHEMBL17242498 0.83 ALDH1A1 (0.51) MAPK1ALDH1A1L3MBTL1KDM4EHPGD
SCHEMBL1065379 0.80 HDAC1 (0.64) MAPK1
SCHEMBL6390385 0.79 MAPK1 (0.46) MAPK1CA12CA9B3GNT2
SCHEMBL25335125 0.78 ALDH1A1 (0.55) MAPK1ALDH1A1L3MBTL1KDM4EHPGD
SCHEMBL31160981 0.78 ALDH1A1 (0.55) MAPK1ALDH1A1L3MBTL1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7868204-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2011-01-11 US disclosed