SCHEMBL10644754

SCHEMBL10644754

NC(=O)CSc1nc2ccccc2o1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.73
RAB9A P51151 5/20 0.69
KMT2A Q03164 3/20 0.69
HPGD P15428 3/20 0.69
MEN1 O00255 2/20 0.69
NPC1 O15118 2/20 0.69
SMN1; SMN2 Q16637 3/20 0.68
TSHR P16473 2/20 0.64
TDP1 Q9NUW8 3/20 0.61
DDAH1 O94760 1/20 0.60
ADRA2C P18825 1/20 0.60
GAA P10253 2/20 0.60
ALPL P05186 1/20 0.60
ALPG P10696 1/20 0.60
POLB P06746 2/20 0.59
MAPT P10636 2/20 0.59
KDM4E B2RXH2 1/20 0.59
USP2 O75604 1/20 0.59
MAPK1 P28482 1/20 0.59
CASP1 P29466 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3500434 0.86 RAB9A (0.76) ALDH1A1RAB9AKMT2AHPGDMEN1
SCHEMBL10403483 0.82 ALDH1A1 (0.69) ALDH1A1RAB9AKMT2AHPGDMEN1
SCHEMBL10403480 0.82 ALDH1A1 (0.69) ALDH1A1RAB9AKMT2AHPGDMEN1
SCHEMBL10402073 0.81 ALDH1A1 (0.68) ALDH1A1RAB9AKMT2AHPGDMEN1
SCHEMBL10402071 0.81 ALDH1A1 (0.68) ALDH1A1RAB9AKMT2AHPGDMEN1
SCHEMBL10644975 0.81 HTT (0.54) ALDH1A1RAB9AKMT2AHPGDMEN1
SCHEMBL10760459 0.81 ALDH1A1 (0.72) ALDH1A1RAB9AKMT2AHPGDMEN1
SCHEMBL14825049 0.79 RAB9A (0.73) ALDH1A1RAB9AKMT2AMEN1NPC1
SCHEMBL12487254 0.79 TSHR (1.00) ALDH1A1RAB9AKMT2AHPGDMEN1
SCHEMBL11275157 0.79 ALDH1A1 (0.72) ALDH1A1RAB9AKMT2AHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009149054-A1 SMALL MOLECULE INHIBITORS FOR THE TREATMENT OR PREVENTION OF DENGUE VIRUS INFECTION SIGA TECHNOLOGIES, INC. (US) 2009-12-10 WO disclosed
US-4719036-A PAINTS; METAL WORKING CIBA-GEIGY CORPORATION (US) 1988-01-12 US disclosed
EP-0006347-B1 COMPOSITIONS AND METHOD FOR REGULATING SOYBEAN PLANT GROWTH UTILIZING SUBSTITUTED BENZAZOLYLTHIOALKANOIC ACIDS MONSANTO COMPANY (US) 1984-01-25 EP disclosed
US-4329363-A Substituted mercapto acid amides and their use MERCK & CO., INC. (US) 1982-05-11 US disclosed