SCHEMBL10649656

SCHEMBL10649656

Cc1[nH]c(-c2cccnc2)nc1C(=O)O

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 7/20 0.72
NPY5R Q15761 3/20 0.58
KMT2A Q03164 1/20 0.54
HPGD P15428 2/20 0.50
DHODH Q02127 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
PKM P14618 1/20 0.50
HCRTR1 O43613 1/20 0.49
CYP1A2 P05177 1/20 0.49
MAPK1 P28482 1/20 0.49
CASP1 P29466 1/20 0.49
CYP2C19 P33261 1/20 0.49
PKN1 Q16512 1/20 0.47
PKN2 Q16513 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10679369 0.88 PIN1 (0.55) PIN1NPY5RKMT2AHPGDKDM4E
SCHEMBL10938735 0.86 PIN1 (0.57) PIN1NPY5RKMT2AHPGDDHODH
SCHEMBL10937913 0.85 PIN1 (0.51) PIN1NPY5RKMT2AHPGDDHODH
SCHEMBL10942001 0.85 PIN1 (0.51) PIN1NPY5RKMT2AHPGDDHODH
SCHEMBL10937354 0.85 PIN1 (0.51) PIN1NPY5RKMT2AHPGDKDM4E
SCHEMBL316552 0.84 PIN1 (1.00) PIN1HPGDKDM4EALDH1A1PKM
SCHEMBL21652629 0.84 PIN1 (0.71) PIN1NPY5RKMT2AHPGDKDM4E
SCHEMBL10679043 0.83 PIN1 (0.50) PIN1NPY5RKMT2AHPGDDHODH
SCHEMBL3418983 0.83 NPY5R (0.50) PIN1NPY5RKMT2AHPGDKDM4E
SCHEMBL10939665 0.82 NPY5R (0.49) PIN1NPY5RKMT2AHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4743586-A PREPARATION FROM A METHYLAMINE, 2-OXIME OF ETHYL 2,3-DIOXOBUTYRATE, HYDRAZINE, TRIETHOXYMETHANE AMERICAN CYANAMID COMPANY (US) 1988-05-10 US disclosed