SCHEMBL10652298

SCHEMBL10652298

CCCCCCCC(=O)Nc1nc(Cl)c2cc[nH]c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 4/20 0.46
HDAC1 Q13547 4/20 0.46
HDAC6 Q9UBN7 4/20 0.46
NPC1 O15118 3/20 0.44
GLA P06280 1/20 0.44
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SPHK2 Q9NRA0 1/20 0.44
SPHK1 Q9NYA1 1/20 0.44
ADORA1 P30542 2/20 0.43
RAB9A P51151 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 2/20 0.41
DEGS1 O15121 1/20 0.41
POLB P06746 1/20 0.41
EP300 Q09472 1/20 0.41
JAK1 P23458 1/20 0.40
XDH P47989 1/20 0.40
CETP P11597 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7160631 0.76 SPHK2 (0.55) JAK2HDAC1HDAC6NPC1SPHK2
SCHEMBL13227316 0.75 KMT2A (0.55) NPC1GLAMAPK1L3MBTL1SPHK2
SCHEMBL13663989 0.74 ADORA1 (0.43) JAK2ADORA1ALDH1A1LMNAJAK1
SCHEMBL9564261 0.73 KMT2A (0.57) NPC1GLAMAPK1L3MBTL1SPHK2
SCHEMBL16351353 0.73 SPHK2 (0.44) JAK2HDAC1HDAC6NPC1GLA
SCHEMBL11016976 0.71 DEGS1 (0.53) NPC1GLAMAPK1L3MBTL1SPHK2
SCHEMBL11018471 0.71 DEGS1 (0.53) NPC1GLAMAPK1L3MBTL1SPHK2
SCHEMBL3626598 0.71 DEGS1 (0.53) NPC1GLAMAPK1L3MBTL1SPHK2
SCHEMBL16351352 0.71 ALDH1A1 (0.42) HDAC1NPC1GLAMAPK1SPHK2
SCHEMBL11015102 0.70 NPC1 (0.51) NPC1GLAMAPK1L3MBTL1SPHK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0119591-B1 THIODEAZAPURINE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 1988-06-22 EP disclosed
US-4595530-A Thiodeazapurine derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1986-06-17 US disclosed
EP-0119591-A1 Thiodeazapurine derivatives Takeda Chemical Industries, Ltd. (JP) 1984-09-26 EP disclosed