SCHEMBL1065307

SCHEMBL1065307

Fc1[c]c(Cl)cc(-c2ccccc2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
ALDH1A1 P00352 5/20 0.38
ESR2 Q92731 1/20 0.35
AKR1C2 P52895 2/20 0.34
AKR1C1 Q04828 2/20 0.34
NPSR1 Q6W5P4 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
HPGD P15428 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
CYP2A6 P11509 1/20 0.32
KDM4E B2RXH2 1/20 0.32
POLB P06746 1/20 0.32
HTT P42858 1/20 0.32
MAOA P21397 1/20 0.31
KIF11 P52732 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1068381 0.84 CYP1A2 (0.48) CYP1A2ALDH1A1ESR2AKR1C2AKR1C1
SCHEMBL1069867 0.84 ALDH1A1 (0.47) CYP1A2ALDH1A1AKR1C2AKR1C1SMN1; SMN2
SCHEMBL27522805 0.82 CYP1A2 (0.46) CYP1A2ALDH1A1ESR2AKR1C2AKR1C1
SCHEMBL4762846 0.79 PTPRC (0.40) ALDH1A1SMN1; SMN2HPGDL3MBTL1PDK2
SCHEMBL6770612 0.79 CYP2A6 (0.47) ALDH1A1MEN1KMT2ASMN1; SMN2TDP1
SCHEMBL15636974 0.76 TTR (0.35) L3MBTL1
SCHEMBL1066310 0.75 ALDH1A1 (0.38) ALDH1A1AKR1C2AKR1C1MEN1KMT2A
SCHEMBL1068489 0.75 CYP1A2 (0.39) CYP1A2ALDH1A1ESR2AKR1C2AKR1C1
SCHEMBL4928553 0.72 KIF11 (0.42) ALDH1A1AKR1C2AKR1C1CRHBPCRHR2
SCHEMBL19953076 0.71 AHR (0.50) CYP1A2ALDH1A1SMN1; SMN2CYP2A6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006886-A2 AZOLE COMPOUNDS CARRYING A SULFUR SUBSTITUENT XIV BASF SE (DE) 2011-01-20 WO disclosed
US-20080318962-A1 Fungicides Based on Nitrogen-Containing Heterocycles SYNGENTA CROP PROTECTION, INC. (US) 2008-12-25 US disclosed
EP-1771423-A1 FUNGICIDES BASED ON NITROGEN-CONTAINING HETEROCYCLES Syngeta Participations AG (CH) 2007-04-11 EP disclosed
WO-2005123698-A1 FUNGICIDES BASED ON NITROGEN-CONTAINING HETEROCYCLES SYNGENTA PARTICIPATIONS AG (CH) 2005-12-29 WO disclosed
EP-1144381-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GmbH (DE) 2001-10-17 EP disclosed
EP-1133475-A1 SUBSTITUTED BENZO DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GmbH (DE) 2001-09-19 EP disclosed
WO-2000032577-A2 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GMBH (DE) 2000-06-08 WO disclosed
WO-2000031039-A1 SUBSTITUTED BENZO[DE]ISOQUINOLINE-1,3-DIONES MERCK PATENT GMBH (DE) 2000-06-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080318962-A1 Fungicides Based on Nitrogen-Containing Heterocycles DDT, CYP4X1, CBR1 CYP1A2 21/4885ALDH1A1 2559/4885ESR2 1563/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.