SCHEMBL10653191

SCHEMBL10653191

COC(=O)C1=C(C)N(O)C(C)=C(C(=O)OC(C)C)C1c1cccc(Cl)c1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 13/20 0.53
PYGM P11217 13/20 0.53
CYP2C9 P11712 5/20 0.53
CYP1A2 P05177 4/20 0.53
CYP3A4 P08684 4/20 0.53
CYP2C19 P33261 4/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
ABCB11 O95342 3/20 0.53
KDM4E B2RXH2 2/20 0.53
HIF1A Q16665 2/20 0.53
HSD17B10 Q99714 2/20 0.53
CYP2D6 P10635 2/20 0.53
NR1I2 O75469 2/20 0.53
NR3C1 P04150 2/20 0.53
ADORA3 P0DMS8 2/20 0.53
TBXA2R P21731 2/20 0.53
OPRK1 P41145 2/20 0.53
SLC6A3 Q01959 2/20 0.53
PDE4D Q08499 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7408943 0.85 CYP2C9 (0.73) CYP2C9CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL7275567 0.83 PYGL (0.49) PYGLPYGMCYP2C9CYP1A2CYP3A4
SCHEMBL7434419 0.78 CYP2C9 (0.61) PYGLPYGMCYP2C9CYP1A2CYP3A4
SCHEMBL7429254 0.78 CYP2C9 (0.64) PYGLPYGMCYP2C9CYP1A2CYP3A4
SCHEMBL7429854 0.78 CYP2C9 (0.61) PYGLPYGMCYP2C9CYP1A2CYP3A4
SCHEMBL7325004 0.78 CYP2C9 (0.64) PYGLPYGMCYP2C9CYP1A2CYP3A4
SCHEMBL8438483 0.77 TSHR (0.60) CYP2C9CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL10476906 0.77 CYP2C9 (0.59) PYGLPYGMCYP2C9CYP1A2CYP3A4
SCHEMBL11451334 0.76 CYP2C9 (0.60) CYP2C9CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL11461372 0.76 CYP2C9 (0.60) CYP2C9CYP1A2CYP3A4CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0093945-B1 1,4-DIHYDROPYRIDINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1988-11-23 EP claimed
US-4495192-A HYPOTENSIVE AGENTS; VASODILATORS KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-22 US claimed
EP-0093945-A2 1,4-Dihydropyridine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1983-11-16 EP claimed
EP-0093945-B1 1,4-DIHYDROPYRIDINE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1988-11-23 EP disclosed
US-4495192-A HYPOTENSIVE AGENTS; VASODILATORS KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-22 US disclosed
EP-0093945-A2 1,4-Dihydropyridine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1983-11-16 EP disclosed