SCHEMBL10657128

SCHEMBL10657128

CSC(SC)=C(C#N)C(=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.65
MAPT P10636 2/20 0.65
XBP1 P17861 2/20 0.65
MAPK1 P28482 2/20 0.65
RAB9A P51151 2/20 0.65
NPSR1 Q6W5P4 2/20 0.65
LMNA P02545 1/20 0.65
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
NPC1 O15118 1/20 0.51
PKM P14618 1/20 0.51
DHODH Q02127 2/20 0.49
GSK3B P49841 2/20 0.42
RAPGEF3 O95398 2/20 0.41
RAPGEF4 Q8WZA2 2/20 0.41
TRPV1 Q8NER1 2/20 0.41
SRD5A2 P31213 1/20 0.40
NR4A1 P22736 1/20 0.40
NR4A2 P43354 1/20 0.40
NR4A3 Q92570 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3129088 0.86 MAPT (0.67) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL7572160 0.83 ALDH1A1 (0.64) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL10651600 0.83 ALDH1A1 (0.71) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL11335661 0.81 DHODH (0.62) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL11335664 0.81 DHODH (0.62) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL10655256 0.81 ALDH1A1 (0.73) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL2443924 0.80 NPSR1 (0.71) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL1416827 0.79 ALDH1A1 (1.00) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL5914784 0.78 CES2 (0.51) ALDH1A1MAPTXBP1MAPK1RAB9A
SCHEMBL5914790 0.78 CES2 (0.51) ALDH1A1MAPTXBP1MAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273602-A1 3-Cyano-4-arylthiophenes ELI LILLY AND COMPANY (US) 1988-07-06 EP disclosed