SCHEMBL10659604

SCHEMBL10659604

COc1cc2c(cc1OC)C(C)N(C(=O)Cc1ccc(OC(C)=O)cc1)CC2

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.71
SMN1; SMN2 Q16637 1/20 0.61
KDM4E B2RXH2 1/20 0.61
TP53 P04637 3/20 0.57
POLB P06746 1/20 0.57
LMNA P02545 3/20 0.55
MAPK1 P28482 1/20 0.55
HTT P42858 1/20 0.55
TSHR P16473 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11291966 0.88 KMT2A (0.57) KMT2ASMN1; SMN2KDM4ETP53POLB
SCHEMBL10661700 0.86 KMT2A (0.76) KMT2ASMN1; SMN2KDM4ETP53POLB
SCHEMBL10661988 0.82 KMT2A (0.70) KMT2ASMN1; SMN2KDM4ETP53POLB
SCHEMBL10660418 0.78 ABCB1 (0.78) KMT2ASMN1; SMN2KDM4EPOLBMAPK1
SCHEMBL11459473 0.78 KMT2A (0.48) KMT2ASMN1; SMN2KDM4ETP53POLB
SCHEMBL22970639 0.77 SMN1; SMN2 (0.71) KMT2ASMN1; SMN2KDM4EPOLBLMNA
SCHEMBL10660441 0.77 SMN1; SMN2 (0.72) KMT2ASMN1; SMN2KDM4EPOLBLMNA
SCHEMBL10662225 0.75 KMT2A (0.64) KMT2ASMN1; SMN2KDM4EPOLBHTT
SCHEMBL10660245 0.73 KMT2A (0.55) KMT2ASMN1; SMN2KDM4EPOLBLMNA
SCHEMBL22782437 0.72 SMN1; SMN2 (0.83) KMT2ASMN1; SMN2KDM4EPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766131-A 2-amino (or hydroxy) phenethyl-1,2,3,4-tetrahydroisoquinolines as analgesics PENNWALT CORPORATION (US) 1988-08-23 US disclosed
EP-0051190-A2 N-(amino(or hydroxy) phenethyl)-1,2,3,4-tetrahydroisoquinolines, precursors thereof, and methods of preparation PENNWALT CORPORATION (US) 1982-05-12 EP disclosed