SCHEMBL10660441

SCHEMBL10660441

COc1cc2c(cc1OC)C(C)N(C(=O)Cc1cccc([N+](=O)[O-])c1)CC2

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.72
HTT P42858 1/20 0.72
NCOA1 Q15788 1/20 0.72
NCOA3 Q9Y6Q9 1/20 0.72
KMT2A Q03164 4/20 0.62
HTR1A P08908 2/20 0.59
HTR1D P28221 2/20 0.59
HTR1B P28222 2/20 0.59
KDM4E B2RXH2 1/20 0.58
MAPT P10636 1/20 0.57
GRIN2C Q14957 1/20 0.56
NPSR1 Q6W5P4 2/20 0.56
LMNA P02545 1/20 0.56
NPC1 O15118 1/20 0.52
POLB P06746 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10661988 0.90 KMT2A (0.70) SMN1; SMN2HTTNCOA1NCOA3KMT2A
Hydrochloric Acid SCHEMBL11286503 0.87 HTT (0.59) SMN1; SMN2HTTNCOA1NCOA3KMT2A
SCHEMBL10662225 0.82 KMT2A (0.64) SMN1; SMN2HTTNCOA1NCOA3KMT2A
SCHEMBL10661700 0.79 KMT2A (0.76) SMN1; SMN2HTTKMT2AKDM4ENPSR1
Hydrochloric Acid SCHEMBL10660995 0.79 HTT (0.62) SMN1; SMN2HTTNCOA1NCOA3KMT2A
SCHEMBL10660245 0.79 KMT2A (0.55) SMN1; SMN2HTTNCOA1NCOA3KMT2A
SCHEMBL10659604 0.77 KMT2A (0.71) SMN1; SMN2HTTKMT2AKDM4ELMNA
SCHEMBL22970639 0.75 SMN1; SMN2 (0.71) SMN1; SMN2HTTKMT2AKDM4ENPSR1
SCHEMBL6604720 0.75 HTR1B (1.00) SMN1; SMN2HTTNCOA1NCOA3HTR1A
SCHEMBL6604715 0.75 HTR1B (1.00) SMN1; SMN2HTTNCOA1NCOA3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766131-A 2-amino (or hydroxy) phenethyl-1,2,3,4-tetrahydroisoquinolines as analgesics PENNWALT CORPORATION (US) 1988-08-23 US disclosed
EP-0051190-A2 N-(amino(or hydroxy) phenethyl)-1,2,3,4-tetrahydroisoquinolines, precursors thereof, and methods of preparation PENNWALT CORPORATION (US) 1982-05-12 EP disclosed