SCHEMBL10661700

SCHEMBL10661700

COc1cc2c(cc1OC)C(C)N(C(=O)Cc1ccc(N)cc1)CC2

nearest known ligand 0.76

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.76
KDM4E B2RXH2 1/20 0.64
SMN1; SMN2 Q16637 2/20 0.61
LMNA P02545 3/20 0.58
HTT P42858 2/20 0.58
MAPK1 P28482 1/20 0.58
TP53 P04637 3/20 0.57
ALDH1A1 P00352 1/20 0.55
GAA P10253 1/20 0.55
TSHR P16473 1/20 0.55
RAB9A P51151 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55
POLB P06746 2/20 0.55
NPC1 O15118 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10659604 0.86 KMT2A (0.71) KMT2AKDM4ESMN1; SMN2LMNAHTT
SCHEMBL10661988 0.85 KMT2A (0.70) KMT2AKDM4ESMN1; SMN2LMNAHTT
SCHEMBL22970639 0.80 SMN1; SMN2 (0.71) KMT2AKDM4ESMN1; SMN2LMNAHTT
SCHEMBL11389038 0.80 KMT2A (0.67) KMT2AKDM4ESMN1; SMN2HTTNPC1
SCHEMBL10660441 0.79 SMN1; SMN2 (0.72) KMT2AKDM4ESMN1; SMN2LMNAHTT
Veradoline SCHEMBL489286 0.76 MAOA (0.53) KMT2AKDM4ESMN1; SMN2LMNAMAPK1
Veradoline SCHEMBL29388371 0.76 MAOA (0.53) KMT2AKDM4ESMN1; SMN2LMNAMAPK1
Hydrochloric Acid SCHEMBL11291966 0.76 KMT2A (0.57) KMT2AKDM4ESMN1; SMN2LMNAHTT
SCHEMBL10662225 0.75 KMT2A (0.64) KMT2AKDM4ESMN1; SMN2HTTALDH1A1
Veradoline SCHEMBL10656736 0.75 MAOA (0.55) KDM4ESMN1; SMN2LMNAMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766131-A 2-amino (or hydroxy) phenethyl-1,2,3,4-tetrahydroisoquinolines as analgesics PENNWALT CORPORATION (US) 1988-08-23 US disclosed
EP-0051190-A2 N-(amino(or hydroxy) phenethyl)-1,2,3,4-tetrahydroisoquinolines, precursors thereof, and methods of preparation PENNWALT CORPORATION (US) 1982-05-12 EP disclosed