SCHEMBL10661985

SCHEMBL10661985

C=CCn1[c]cc(=O)cc1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.35
CASP3 P42574 2/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CA12 O43570 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
NPC1 O15118 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9798176 0.69 CYP3A4 (0.42) CYP3A4CASP3CYP1A2CYP2D6CA12
SCHEMBL6605535 0.65 CYP3A4 (0.32) CYP3A4CYP1A2CYP2D6
SCHEMBL849669 0.64
SCHEMBL6599824 0.64
SCHEMBL9656980 0.60
SCHEMBL6675403 0.58 CYP3A4 (0.52) CYP3A4CASP3CYP1A2CYP2D6GAA
SCHEMBL9292715 0.58 CYP3A4 (0.35) CYP3A4CYP1A2CYP2D6GAANPC1
SCHEMBL6028160 0.58 CYP3A4 (0.50) CYP3A4CYP1A2CYP2D6GAAKMT2A
SCHEMBL10664405 0.58 CYP3A4 (0.35) CYP3A4CASP3CA12CA2CA9
SCHEMBL9292277 0.58 CASP3 (0.38) CYP3A4CASP3CA12CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4727076-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LTD. (GB) 1988-02-23 US disclosed